SCHEMBL764305

SCHEMBL764305

Cc1ccc(-c2ccc(C(=O)NCCO)cc2)s1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.58
KDM4E B2RXH2 1/20 0.58
PRF1 P14222 2/20 0.52
MMP13 P45452 1/20 0.51
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
NPSR1 Q6W5P4 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
NEK1 Q96PY6 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
POLB P06746 3/20 0.44
HPGD P15428 1/20 0.44
HTT P42858 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24343521 0.88 KDM4E (0.49) ALDH1A1KDM4ENPSR1L3MBTL1POLB
SCHEMBL2021463 0.80 PRF1 (0.61) ALDH1A1KDM4EPRF1MMP13CA12
SCHEMBL24534467 0.80 NPC1 (0.51) ALDH1A1KDM4EPRF1MMP13HDAC6
SCHEMBL17921126 0.78 NPC1 (0.41) ALDH1A1KDM4EPRF1CA12CA1
SCHEMBL620074 0.77 POLB (0.66) ALDH1A1KDM4EMMP13CA12CA1
SCHEMBL17921131 0.77 MAPT (0.39) ALDH1A1KDM4ECA1CA2L3MBTL1
SCHEMBL23110055 0.77 ACKR3 (0.62) ALDH1A1KDM4EMMP13HPGDNPC1
SCHEMBL764574 0.76 MMP13 (0.81) ALDH1A1KDM4EMMP13CA12CA1
SCHEMBL16250219 0.75 NPC1 (0.55) ALDH1A1KDM4EMMP13L3MBTL1HDAC6
SCHEMBL16511794 0.75 SLC6A2 (0.45) MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078015-B1 MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1 AND/OR NF-KAPPAB ACTIVITY AND USE THEREOF BRISTOL MYERS SQUIBB CO (US) 2012-03-21 EP disclosed