SCHEMBL764500

SCHEMBL764500

CC(O)c1ccc(Oc2ccc(CNC(=O)C3(NC(=O)c4ccccc4)CC3)cc2)c(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 2/20 0.43
MAPK14 Q16539 5/20 0.43
EPHX2 P34913 1/20 0.39
CTSL P07711 1/20 0.39
CTSK P43235 1/20 0.39
PSMB11 A5LHX3 1/20 0.38
PSMA7 O14818 1/20 0.38
PSMB1 P20618 1/20 0.38
PSMA1 P25786 1/20 0.38
PSMA2 P25787 1/20 0.38
PSMA3 P25788 1/20 0.38
PSMA4 P25789 1/20 0.38
PSMB8 P28062 1/20 0.38
PSMB9 P28065 1/20 0.38
PSMA5 P28066 1/20 0.38
PSMB4 P28070 1/20 0.38
PSMB6 P28072 1/20 0.38
PSMB5 P28074 1/20 0.38
PSMB10 P40306 1/20 0.38
PSMB3 P49720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13165713 0.94 MAPK14 (0.40) BDKRB1MAPK14EPHX2CTSLCTSK
SCHEMBL13166110 0.91 MAPK14 (0.39) BDKRB1MAPK14EPHX2CTSLHPGD
SCHEMBL10121335 0.90 BDKRB1 (0.45) BDKRB1HPGDSCN9A
SCHEMBL765640 0.89 SCN9A (0.38) BDKRB1MAPK14PSMB11PSMA7PSMB1
SCHEMBL764425 0.89 BDKRB1 (0.48) BDKRB1MAPK14PSMB11PSMA7PSMB1
SCHEMBL765827 0.88 BDKRB1 (0.39) BDKRB1MAPK14PSMB11PSMA7PSMB1
SCHEMBL12238931 0.88 EPHX2 (0.53) BDKRB1MAPK14EPHX2CTSL
SCHEMBL765568 0.87 SCN9A (0.37) BDKRB1MAPK14PSMB11PSMA7PSMB1
SCHEMBL13904206 0.86 BDKRB1 (0.39) BDKRB1PSMB11PSMA7PSMB1PSMA1
SCHEMBL13165586 0.86 BDKRB1 (0.41) BDKRB1HPGDSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188254-B1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-03-21 EP disclosed