SCHEMBL764562

SCHEMBL764562

O=C(NC1CCCCC1)C1Cc2cc(Cl)ccc2N1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.47
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
NPC1 O15118 4/20 0.45
EPHX1 P07099 3/20 0.44
CYP2C19 P33261 2/20 0.44
ALDH1A1 P00352 2/20 0.44
POLB P06746 1/20 0.44
CYP2C9 P11712 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ALOX12 P18054 1/20 0.44
EPHX2 P34913 3/20 0.43
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.43
TSHR P16473 1/20 0.43
CYP1A2 P05177 1/20 0.43
MAPK1 P28482 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HPGD P15428 1/20 0.43
ALOX15 P16050 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL764531 0.81 SMYD3 (0.40) RAB9AMEN1KMT2ANPC1EPHX1
SCHEMBL10280029 0.79 CCR1 (0.39) MEN1KMT2AALDH1A1EPHX2L3MBTL1
SCHEMBL3256484 0.76 GAA (0.60) MAPT
SCHEMBL6246219 0.76 GAA (0.60) MAPT
SCHEMBL6164822 0.76 GAA (0.60) MAPT
SCHEMBL13889887 0.75 GAA (0.42) ALDH1A1MAPTCYP1A2HPGD
SCHEMBL1760636 0.75 SIRT1 (0.44) MAPT
Hydrochloric Acid SCHEMBL11071035 0.75 GAA (0.58) MAPT
Water SCHEMBL28741688 0.75 GAA (0.58) MAPT
SCHEMBL3256076 0.74 PDE5A (0.41) MEN1KMT2AALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1270557-B1 ETHYLENEDIAMINE DERIVATIVES DAIICHI SANKYO CO LTD (JP) 2012-07-25 EP disclosed
EP-2431370-A1 Monoacylated 1,2-diaminocycloalkanes DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2012-03-21 EP disclosed