SCHEMBL7647

SCHEMBL7647

O=C(O)c1nc2cccc(O)c2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.42
KDM4E B2RXH2 4/20 0.41
TDP1 Q9NUW8 2/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
GUSB P08236 2/20 0.41
HPGD P15428 1/20 0.41
ACHE P22303 1/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
AURKA O14965 1/20 0.38
DYRK1A Q13627 4/20 0.36
PARP1 P09874 2/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4629095 0.84 PIM1 (0.40) KDM4ETDP1GUSBHPGDACHE
SCHEMBL8952892 0.82 ALDH1A1 (0.47) PIN1KDM4ETDP1HPGDALDH1A1
SCHEMBL7706759 0.81 DYRK1A (0.51) PIN1KDM4ECA12CA9GUSB
SCHEMBL6961429 0.81 PIN1 (0.41) PIN1KDM4ETDP1HPGDKMT2A
SCHEMBL30310472 0.81 DYRK1A (0.51) PIN1KDM4ECA12CA9GUSB
SCHEMBL6988205 0.81 DYRK1A (0.42) PIN1CA12CA9ALDH1A1MAPT
SCHEMBL1144716 0.81 PIN1 (0.49) PIN1KDM4EHPGDKMT2AALDH1A1
SCHEMBL11047670 0.81 PIN1 (0.41) PIN1KDM4ETDP1HPGDALDH1A1
SCHEMBL11195012 0.78 PARP1 (0.43) KDM4ETDP1GUSBHPGDKMT2A
SCHEMBL31569165 0.78 PIN1 (0.40) PIN1KDM4ETDP1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499114-A1 COMPOUNDS INHIBITORS OF ENZYME LACTATE DEHYDROGENASE (LDH) AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS Universita Di Pisa (IT) 2012-09-19 EP disclosed
WO-2011054525-A1 COMPOUNDS INHIBITORS OF ENZYME LACTATE DEHYDROGENASE (LDH) AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS UNIVERSITA' DI PISA (IT) 2011-05-12 WO disclosed