SCHEMBL7649136

SCHEMBL7649136

CCCCCCc1cc2c(cc1C#Cc1ccc(CC(=O)O)cc1)C(CC)(CC)CCO2

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
CYP26A1 O43174 1/20 0.36
CYP26B1 Q9NR63 1/20 0.36
FFAR1 O14842 4/20 0.36
FFAR4 Q5NUL3 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PLA2G4B P0C869 1/20 0.34
RARB P10826 1/20 0.33
RARG P13631 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
PTPN11 Q06124 3/20 0.32
PTPN1 P18031 1/20 0.32
PTPN6 P29350 1/20 0.32
PTGER4 P35408 2/20 0.31
PTPRO Q16827 1/20 0.31
ACACB O00763 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7651242 0.90 FFAR1 (0.40) CYP26A1CYP26B1FFAR1FFAR4ACACB
SCHEMBL8662753 0.90 FDFT1 (0.36) FFAR1FFAR4THRATHRB
SCHEMBL7653907 0.87 ALDH1A1 (0.34) ALDH1A1CYP26A1CYP26B1FFAR1FFAR4
SCHEMBL7652608 0.86 PTGDR2 (0.33) PTGDR2
SCHEMBL8673367 0.85 CYP4F2 (0.35) FFAR1FFAR4THRATHRB
SCHEMBL7653071 0.84 FFAR1 (0.32) FFAR1
SCHEMBL7654470 0.84 MAPT (0.36) ALDH1A1HPGDHSD17B10RARBRARG
SCHEMBL7660646 0.84 FFAR1 (0.40) CYP26A1CYP26B1FFAR1FFAR4ACACB
SCHEMBL7655942 0.83 PTGDR2 (0.31) PTGDR2
SCHEMBL7656413 0.81 PTGDR2 (0.34) PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344463-B1 SKIN DISORDERS, ACNE ALLERGAN SALES, INC. 2002-02-05 US disclosed
EP-0636127-B1 Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN INC (US) 2001-04-04 EP disclosed
US-6090826-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN SALES, INC. (US) 2000-07-18 US disclosed
US-5663347-A REGULATORS OF CELL PROLIFERATION AND DIFFERENTIATION; TREATMENT OF SKIN DISORDERS; ANTICARCINOGNIC AGENTS ALLERGAN (US) 1997-09-02 US disclosed
US-5468879-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN, INC. (US) 1995-11-21 US disclosed
EP-0636127-A1 DISUBSTITUTED ACETYLENES BEARING HETEROBICYCLIC GROUPS AND HETEROAROMATIC OR PHENYL GROUPS HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC. (US) 1995-02-01 EP disclosed
WO-1993016068-A1 DISUBSTITUTED ACETYLENES BEARING HETEROBICYCLIC GROUPS AND HETEROAROMATIC OR PHENYL GROUPS HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC. (US) 1993-08-19 WO disclosed