SCHEMBL7653907

SCHEMBL7653907

CCCCCCc1cc2c(cc1C#Cc1ccc(CC(=O)O)cn1)C(CC)(CC)CCO2

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.33
CYP26A1 O43174 1/20 0.32
CYP26B1 Q9NR63 1/20 0.32
FFAR1 O14842 1/20 0.32
FFAR4 Q5NUL3 1/20 0.32
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31
RARB P10826 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6664722 0.91 CYP26A1 (0.41) ALDH1A1PTGDR2CYP26A1CYP26B1FFAR1
SCHEMBL7652436 0.91 CYP26A1 (0.35) PTGDR2CYP26A1CYP26B1FFAR1FFAR4
SCHEMBL8661568 0.91 CYP3A4 (0.33) PTGDR2RARB
SCHEMBL7656413 0.88 PTGDR2 (0.34) PTGDR2
SCHEMBL7649136 0.87 ALDH1A1 (0.40) ALDH1A1PTGDR2CYP26A1CYP26B1FFAR1
SCHEMBL7652859 0.87 CYP3A4 (0.33) PTGDR2FFAR1FFAR4RARB
SCHEMBL7655942 0.87 PTGDR2 (0.31) PTGDR2
SCHEMBL7651528 0.85 CYP26A1 (0.35) PTGDR2CYP26A1CYP26B1FFAR1FFAR4
SCHEMBL8147495 0.85 ALOX5 (0.35) ALDH1A1PTGDR2
SCHEMBL7652366 0.85 KMT2A (0.44) ALDH1A1PTGDR2CYP26A1HSD17B10RARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344463-B1 SKIN DISORDERS, ACNE ALLERGAN SALES, INC. 2002-02-05 US disclosed
EP-0636127-B1 Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN INC (US) 2001-04-04 EP disclosed
US-5663347-A REGULATORS OF CELL PROLIFERATION AND DIFFERENTIATION; TREATMENT OF SKIN DISORDERS; ANTICARCINOGNIC AGENTS ALLERGAN (US) 1997-09-02 US disclosed
US-5468879-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN, INC. (US) 1995-11-21 US disclosed
EP-0636127-A1 DISUBSTITUTED ACETYLENES BEARING HETEROBICYCLIC GROUPS AND HETEROAROMATIC OR PHENYL GROUPS HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC. (US) 1995-02-01 EP disclosed
US-5264578-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN, INC. (US) 1993-11-23 US disclosed
WO-1993016068-A1 DISUBSTITUTED ACETYLENES BEARING HETEROBICYCLIC GROUPS AND HETEROAROMATIC OR PHENYL GROUPS HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC. (US) 1993-08-19 WO disclosed