SCHEMBL7650151

SCHEMBL7650151

CC(C)c1ccc(C(=O)Nc2ccc3c(c2)CN(C)CC3(C)C)cc1S(=O)(=O)C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDR1 Q08345 1/20 0.40
DDR2 Q16832 1/20 0.40
MAPT P10636 5/20 0.38
LMNA P02545 2/20 0.38
TP53 P04637 1/20 0.37
ROCK2 O75116 4/20 0.37
RAB9A P51151 4/20 0.36
RARA P10276 3/20 0.36
RARB P10826 3/20 0.36
RARG P13631 3/20 0.36
NPC1 O15118 3/20 0.36
ALDH1A1 P00352 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 2/20 0.36
CYP26A1 O43174 2/20 0.36
CYP3A4 P08684 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7653759 0.82 ROCK2 (0.42) DDR1DDR2ROCK2RAB9ARARA
SCHEMBL7993332 0.80 ROCK2 (0.45) DDR1DDR2ROCK2RARARARB
SCHEMBL7652080 0.76 DDR1 (0.43) DDR1DDR2MAPTTP53ROCK2
SCHEMBL7652898 0.76 KIT (0.49) DDR1DDR2EGFRBRAF
Hydrochloric Acid SCHEMBL7657621 0.76 DDR1 (0.42) DDR1DDR2MAPTTP53ROCK2
SCHEMBL7989876 0.75 MAPT (0.47) MAPTTP53ROCK2RAB9ANPC1
Hydrochloric Acid SCHEMBL7658653 0.75 KIT (0.48) DDR1DDR2EGFRBRAF
SCHEMBL7653791 0.75 MAPT (0.45) DDR1DDR2MAPTLMNATP53
SCHEMBL6295053 0.74 ROCK2 (0.52) MAPTLMNAROCK2RAB9ANPC1
SCHEMBL7649723 0.74 NPC1 (0.52) DDR1DDR2MAPTROCK2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed