SCHEMBL7652080

SCHEMBL7652080

CC(C)Oc1ccc(C(=O)Nc2ccc3c(c2)CN(C)CC3(C)C)cc1C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDR1 Q08345 1/20 0.43
DDR2 Q16832 1/20 0.43
ROCK2 O75116 4/20 0.42
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42
TP53 P04637 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
THRB P10828 1/20 0.41
BRAF P15056 2/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
RAB9A P51151 1/20 0.40
RAF1 P04049 1/20 0.40
HTR1D P28221 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7657621 0.99 DDR1 (0.42) DDR1DDR2ROCK2MAPTKDM4E
SCHEMBL7989876 0.92 MAPT (0.47) ROCK2MAPTKDM4EMEN1CYP2D6
SCHEMBL7653791 0.89 MAPT (0.45) DDR1DDR2ROCK2MAPTKDM4E
SCHEMBL7993309 0.86 ROCK2 (0.52) ROCK2MAPTKDM4EMEN1HTT
SCHEMBL7661417 0.86 ROCK2 (0.44) DDR1DDR2ROCK2MAPTMEN1
SCHEMBL7649761 0.86 MAPT (0.46) ROCK2MAPTMEN1KMT2ATP53
SCHEMBL6298344 0.86 ROCK2 (0.56) ROCK2MAPTTP53SMN1; SMN2THRB
SCHEMBL7652898 0.85 KIT (0.49) DDR1DDR2BRAFKIT
SCHEMBL7652847 0.84 ROCK2 (0.46) DDR1DDR2ROCK2MAPTKDM4E
SCHEMBL7653787 0.84 ROCK2 (0.43) DDR1DDR2ROCK2MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed