SCHEMBL7650189

SCHEMBL7650189

C[C@H]1CN(c2ccc(C(=O)NCCC(=O)ONC(=O)OCc3ccccc3)cc2)CCN1c1ncccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
HTT P42858 1/20 0.42
HDAC1 Q13547 5/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC3 O15379 1/20 0.41
CYP2C9 P11712 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
MAPKAPK3 Q16644 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
SLC6A7 Q99884 2/20 0.40
FLT1 P17948 2/20 0.38
KDR P35968 2/20 0.38
FLT3 P36888 2/20 0.38
AURKA O14965 1/20 0.38
GAA P10253 1/20 0.38
CHRM4 P08173 2/20 0.37
CASR P41180 1/20 0.37
MAPT P10636 2/20 0.37
AOC3 Q16853 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7655291 0.88 KDM4E (0.53) KDM4EHTTSLC6A7FLT1KDR
SCHEMBL7652415 0.83 KDM4E (0.44) KDM4EHTTSLC6A7CHRM4CASR
SCHEMBL7653652 0.83 KDM4E (0.44) KDM4EHTTSLC6A7CHRM4CASR
SCHEMBL7652041 0.83 KDM4E (0.44) KDM4EHTTSLC6A7CHRM4CASR
SCHEMBL7655338 0.82 ITGB3 (0.49) SLC6A7
SCHEMBL7052907 0.81 ITGB3 (0.40) KDM4EHTTFLT1KDRFLT3
SCHEMBL382409 0.80 KDM4E (0.40) KDM4EHTTGAACHRM4CASR
SCHEMBL7662184 0.78 KDM4E (0.46) KDM4EHTTSLC6A7GAAMAPT
SCHEMBL7650186 0.76 ITGB3 (0.47)
SCHEMBL7654976 0.72 KDM4E (0.44) KDM4EHTTCHRM4MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US claimed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP claimed
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US disclosed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP disclosed