SCHEMBL7651979

SCHEMBL7651979

N=C(N)N1CCN(c2ccc(C(=O)NC(CC(=O)O)NS(=O)(=O)c3ccccc3)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.47
ITGA2B P08514 3/20 0.47
F2 P00734 5/20 0.42
F10 P00742 5/20 0.42
PRSS1 P07477 2/20 0.42
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
ALOX15 P16050 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PKM P14618 1/20 0.41
PLG P00747 3/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CCR1 P32246 1/20 0.40
PLAU P00749 2/20 0.40
ST14 Q9Y5Y6 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7651526 0.85 ITGB3 (0.45) ITGB3ITGA2BALDH1A1PLAUITGAV
SCHEMBL7654428 0.83 ITGB3 (0.48) ITGB3ITGA2BLMNAALDH1A1PKM
SCHEMBL7658155 0.83 MEN1 (0.51) ITGB3ITGA2BUSP2LMNAALOX15
SCHEMBL7651971 0.81 ITGB3 (0.72) ITGB3ITGA2BITGAV
SCHEMBL382764 0.79 ITGB3 (0.51) ITGB3ITGA2BMAPTITGAV
SCHEMBL27551456 0.79 ITGB3 (0.51) ITGB3ITGA2BMAPTITGAV
SCHEMBL7651229 0.79 TP53 (0.46) ITGB3ITGA2BMAPTITGAV
SCHEMBL7651202 0.78 ITGB3 (0.53) ITGB3ITGA2BLMNAALDH1A1PKM
SCHEMBL415668 0.76 DRD4 (0.54) ITGB3ITGA2BALDH1A1
SCHEMBL382937 0.76 ITGB3 (0.66) ITGB3ITGA2BITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US claimed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP claimed
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US disclosed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP disclosed