SCHEMBL7653787

SCHEMBL7653787

CC(C)Oc1ccc(C(=O)Nc2ccc3c(c2)CN(C)CC3(C)C)cc1C(=O)C(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 6/20 0.43
ALDH1A1 P00352 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
TP53 P04637 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP3A4 P08684 3/20 0.40
KCNQ3 O43525 1/20 0.39
KCNQ2 O43526 1/20 0.39
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
HTR2A P28223 1/20 0.38
POLB P06746 1/20 0.38
KCNK3 O14649 1/20 0.38
KCNK9 Q9NPC2 1/20 0.38
RARA P10276 3/20 0.38
RARB P10826 3/20 0.38
RARG P13631 3/20 0.38
MAPK1 P28482 2/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7662369 0.93 ROCK2 (0.49) ROCK2ALDH1A1NPC1RAB9ATP53
SCHEMBL7661417 0.92 ROCK2 (0.44) ROCK2ALDH1A1NPC1RAB9ATP53
SCHEMBL7658055 0.90 MAPT (0.45) ROCK2NPC1RAB9ATP53SMN1; SMN2
SCHEMBL7655617 0.89 ROCK2 (0.42) ROCK2ALDH1A1NPC1RAB9ATP53
SCHEMBL7653708 0.88 ROCK2 (0.40) ROCK2NPC1RAB9ATP53SMN1; SMN2
SCHEMBL7649761 0.87 MAPT (0.46) ROCK2ALDH1A1NPC1RAB9ATP53
SCHEMBL7993309 0.87 ROCK2 (0.52) ROCK2ALDH1A1NPC1RAB9ATP53
SCHEMBL7652080 0.84 DDR1 (0.43) ROCK2ALDH1A1NPC1RAB9ATP53
SCHEMBL7655775 0.84 ROCK2 (0.46) ROCK2ALDH1A1NPC1RAB9ATP53
Hydrochloric Acid SCHEMBL7657621 0.83 DDR1 (0.42) ROCK2ALDH1A1NPC1RAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed