SCHEMBL7652475

SCHEMBL7652475

CN1[C@@H]2CC[C@H]1CC(OC(=O)c1ccccc1C(=O)OC1C[C@H]3CC[C@@H](C1)N3C)C2

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 6/20 0.75
HTR3E A5X5Y0 4/20 0.75
HTR3B O95264 4/20 0.75
HTR3D Q70Z44 4/20 0.75
HTR3C Q8WXA8 4/20 0.75
CHRNA7 P36544 2/20 0.75
CHRM5 P08912 2/20 0.69
CHRM1 P11229 2/20 0.69
CHRM3 P20309 2/20 0.69
CYP2D6 P10635 2/20 0.69
LMNA P02545 2/20 0.69
CHRNA1 P02708 1/20 0.69
CHRNG P07510 1/20 0.69
CYP3A4 P08684 1/20 0.69
HTR1A P08908 1/20 0.69
MAPT P10636 1/20 0.69
CHRNB1 P11230 1/20 0.69
CHRNB2 P17787 1/20 0.69
ADRA2B P18089 1/20 0.69
ADRA2C P18825 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7652481 1.00 HTR3A (0.75) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL5789144 0.94 HTR3A (0.68) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL5789139 0.94 HTR3A (0.68) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL6507170 0.90 HTR3E (0.66) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL5789101 0.90 HTR3A (0.66) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL6507167 0.90 HTR3E (0.66) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL5789103 0.90 HTR3A (0.66) HTR3AHTR3EHTR3BHTR3DHTR3C
Benzoyl Tropine SCHEMBL221830 0.86 HTR3E (1.00) HTR3AHTR3EHTR3BHTR3DHTR3C
Benzoyl Tropine SCHEMBL30954638 0.86 HTR3E (1.00) HTR3AHTR3EHTR3BHTR3DHTR3C
Benzoyl Tropine SCHEMBL1103723 0.86 HTR3E (1.00) HTR3AHTR3EHTR3BHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6376510-B1 ADMINISTERING A ALKOXY- AND ACYLOXY-SUBSTITUTED ARALKYL AND ARALKENYL BIS QUATERNARY AMMONIUM DERIVATIVES OF CYCLIC ALKANOL DIESTERS TO A HUMAN AS MUSCLE RELAXANTS NEWLAXANT LLC 2002-04-23 US disclosed
US-6274757-B1 REACTING AN HYDROXY AMINE CORRESPONDING COMPOUND WITH DICHLORO COMPOUND NEWLAXANT LLC 2001-08-14 US disclosed