SCHEMBL7652750

SCHEMBL7652750

COc1ccc2c(OCC(=O)[C@](N)(CCCNC(=N)N)C(=O)O)cccc2c1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 13/20 0.40
MTNR1B P49286 7/20 0.40
CYP2D6 P10635 1/20 0.40
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
POLB P06746 1/20 0.39
NQO2 P16083 2/20 0.36
AURKA O14965 1/20 0.36
MET P08581 1/20 0.36
KDR P35968 1/20 0.36
TEK Q02763 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
KDM4E B2RXH2 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7652741 0.79 C3AR1 (0.44) MTNR1AMTNR1BCYP2D6ALDH1A1HPGD
SCHEMBL7859245 0.73 NCEH1 (0.36) MTNR1AALDH1A1HPGDPOLBKDM4E
SCHEMBL28216506 0.67 SPHK1 (0.35) ALDH1A1
SCHEMBL27083150 0.67 SPHK1 (0.35) ALDH1A1
SCHEMBL7648460 0.66 C3AR1 (0.53) ALDH1A1HPGDPOLBKDM4ETDP1
SCHEMBL7648470 0.66 C3AR1 (0.53) ALDH1A1HPGDPOLBKDM4ETDP1
SCHEMBL27751170 0.66 ALOX15 (0.40)
SCHEMBL27626286 0.65 SMN1; SMN2 (0.38) POLBTDP1
SCHEMBL5277223 0.65 SMN1; SMN2 (0.38) POLBTDP1
Naphthylamine SCHEMBL27819026 0.64 CYP3A4 (0.36) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6489339-B1 C3A receptor ligands SMITHKLINE BEECHAM CORPORATION 2002-12-03 US claimed
EP-1119357-A1 C3A RECEPTOR LIGANDS SmithKline Beecham Corporation (US) 2001-08-01 EP claimed
WO-2000009129-A1 C3A RECEPTOR LIGANDS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-24 WO claimed
US-6489339-B1 C3A receptor ligands SMITHKLINE BEECHAM CORPORATION 2002-12-03 US disclosed
EP-1119357-A1 C3A RECEPTOR LIGANDS SmithKline Beecham Corporation (US) 2001-08-01 EP disclosed
WO-2000009129-A1 C3A RECEPTOR LIGANDS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-24 WO disclosed