SCHEMBL765302

SCHEMBL765302

CN1CCc2sc(C(N)=O)cc2C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.51
PARP1 P09874 4/20 0.50
PARP2 Q9UGN5 4/20 0.50
PRMT5 O14744 1/20 0.47
WDR77 Q9BQA1 1/20 0.47
HDAC6 Q9UBN7 3/20 0.46
F10 P00742 1/20 0.46
ALDH1A1 P00352 3/20 0.46
HPGD P15428 2/20 0.46
KDM4E B2RXH2 2/20 0.46
MAPT P10636 2/20 0.46
MEN1 O00255 1/20 0.46
GLA P06280 1/20 0.46
KMT2A Q03164 1/20 0.46
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
TP53 P04637 1/20 0.40
MAPK1 P28482 1/20 0.40
NOTUM Q6P988 1/20 0.40
F2 P00734 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3313449 0.86 ALDH1A1 (0.56) PARP1PARP2PRMT5WDR77HDAC6
SCHEMBL12922699 0.82 HDAC6 (0.53) PARP1PARP2PRMT5WDR77HDAC6
SCHEMBL3310243 0.79 KDM4E (0.48) PRMT5WDR77HDAC6F10ALDH1A1
SCHEMBL3309101 0.76 ALDH1A1 (0.64) PNMTPRMT5WDR77HDAC6ALDH1A1
SCHEMBL6421478 0.76 NR1H2 (0.54) PNMTHDAC6KDM4EMAPTNPC1
SCHEMBL25796678 0.74 PARP1 (0.42) PARP1PARP2PRMT5WDR77HDAC6
SCHEMBL29972349 0.74 PNMT (0.44) PNMTPRMT5WDR77HDAC6NPC1
SCHEMBL2761887 0.73 ALDH1A1 (0.56) PARP1PARP2PRMT5WDR77HDAC6
SCHEMBL10513283 0.73 WDR91 (0.50) PNMTPARP1PARP2PRMT5WDR77
SCHEMBL2461710 0.73 ALDH1A1 (0.70) PNMTALDH1A1HPGDMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1405852-B1 DIAMINE DERIVATIVES DAIICHI SANKYO CO LTD (JP) 2012-08-01 EP disclosed
EP-1270557-B1 ETHYLENEDIAMINE DERIVATIVES DAIICHI SANKYO CO LTD (JP) 2012-07-25 EP disclosed
EP-2431370-A1 Monoacylated 1,2-diaminocycloalkanes DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2012-03-21 EP disclosed