SCHEMBL7653146

SCHEMBL7653146

NCCC(c1ccccc1)C(N)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 2/20 0.50
CYP2D6 P10635 2/20 0.47
MEN1 O00255 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
KMT2A Q03164 1/20 0.47
SLC1A2 P43004 2/20 0.44
SLC1A3 P43003 1/20 0.44
SLC1A1 P43005 1/20 0.44
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
HTR2A P28223 1/20 0.42
GRM2 Q14416 2/20 0.42
GRM3 Q14832 2/20 0.42
SRC P12931 1/20 0.42
GABBR2 O75899 1/20 0.42
GABBR1 Q9UBS5 1/20 0.42
DPP4 P27487 2/20 0.41
TAAR1 Q96RJ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5565838 0.87 CYP2D6 (0.46) CYP2D6MEN1CYP2C9CYP2C19KMT2A
SCHEMBL5291382 0.85 SLC6A2 (0.55) CYP2D6MEN1CYP2C9CYP2C19KMT2A
SCHEMBL14842376 0.85 SLC6A2 (0.55) CYP2D6MEN1CYP2C9CYP2C19KMT2A
SCHEMBL22190041 0.85 SLC6A2 (0.55) CYP2D6MEN1CYP2C9CYP2C19KMT2A
SCHEMBL5320862 0.84 CYP2D6 (0.46) CYP2D6MEN1CYP2C9CYP2C19KMT2A
SCHEMBL5283024 0.82 SLC1A3 (0.50) CYP2D6MEN1CYP2C9CYP2C19KMT2A
SCHEMBL5289685 0.81 POLB (0.48) CYP2D6MEN1CYP2C9CYP2C19KMT2A
SCHEMBL6533633 0.80 CSNK1E (0.44) CYP2D6MEN1CYP2C9CYP2C19KMT2A
SCHEMBL17476729 0.80 RIPK1 (0.53) CYP2D6MEN1CYP2C9CYP2C19KMT2A
SCHEMBL497730 0.79 CYP2C19 (0.72) CYP2D6MEN1CYP2C9CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358978-B1 FOR THERAPY AND PROPHYLAXIS OF RHEUMATOID ARTHRITIS (IN THE CASE OF INFLAMMATION), OSTEOARTHRITIS, ASTHMA, CARDIAC INFARCT, ALZHEIMER'S DISEASE, OR ATHEROSCLEROSIS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-03-19 US disclosed