SCHEMBL7653165

SCHEMBL7653165

CC(C)(C)OC(=O)C(CNC(=O)c1ccc(N2CCN(c3ncccn3)CC2)cc1)NCS(=O)(=O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.45
ITGA2B P08514 3/20 0.45
GAA P10253 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
ITGAV P06756 2/20 0.40
HTT P42858 2/20 0.40
KDM4E B2RXH2 1/20 0.40
SMN1; SMN2 Q16637 4/20 0.39
MEN1 O00255 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MAPT P10636 2/20 0.38
LMNA P02545 2/20 0.38
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7651421 0.90 ITGB3 (0.42) ITGB3ITGA2BGAANPC1RAB9A
SCHEMBL7649706 0.88 ITGB3 (0.55) ITGB3ITGA2BGAANPC1RAB9A
SCHEMBL7653161 0.82 ITGB3 (0.42) ITGB3ITGA2BNPC1RAB9ACA1
SCHEMBL7652521 0.78 ITGB3 (0.51) ITGB3ITGA2BNPC1RAB9ACA1
SCHEMBL7654405 0.77 ITGB3 (0.74) ITGB3ITGA2BITGAV
SCHEMBL7651416 0.77 ITGB3 (0.38) ITGB3ITGA2BNPC1RAB9ACA1
SCHEMBL7653684 0.75 ITGB3 (0.70) ITGB3ITGA2BITGAV
SCHEMBL383058 0.74 ITGB3 (0.58) ITGB3ITGA2BITGAV
SCHEMBL7649732 0.73 ITGB3 (0.48) ITGB3ITGA2BGAANPC1RAB9A
SCHEMBL7655259 0.73 ITGB3 (0.59) ITGB3ITGA2BITGAVMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US claimed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP claimed
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US disclosed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP disclosed