SCHEMBL7653286

SCHEMBL7653286

COC(=O)c1c(-c2ccc(Cl)cc2)[nH]c2ccccc12

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.68
ALOX5 P09917 4/20 0.67
CCNB2 O95067 1/20 0.52
CDK1 P06493 1/20 0.52
CCNB1 P14635 1/20 0.52
CCNB3 Q8WWL7 1/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
KDM4E B2RXH2 1/20 0.52
ALDH1A1 P00352 1/20 0.52
HPGD P15428 1/20 0.52
HSD17B10 Q99714 1/20 0.52
LMNA P02545 1/20 0.52
MAPT P10636 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5438097 0.88 NR4A2 (0.69) NR4A2ALOX5MEN1KMT2AKDM4E
SCHEMBL14709940 0.85 NR4A2 (0.61) NR4A2ALOX5MEN1KMT2AKDM4E
SCHEMBL31312750 0.85 TUBB4A (0.62) NR4A2ALOX5MEN1KMT2AKDM4E
SCHEMBL5621441 0.84 NR4A2 (0.60) NR4A2ALOX5MEN1KMT2AKDM4E
SCHEMBL6492107 0.83 CCNB2 (0.56) ALOX5CCNB2CDK1CCNB1CCNB3
SCHEMBL5137730 0.81 NR4A2 (1.00) NR4A2ALOX5MEN1KMT2AKDM4E
SCHEMBL4338589 0.81 ALOX5 (1.00) NR4A2ALOX5MEN1KMT2AKDM4E
SCHEMBL18180604 0.80 CCNB2 (0.53) CCNB2CDK1CCNB1CCNB3MEN1
SCHEMBL31312633 0.80 ALOX5 (0.57) NR4A2ALOX5
SCHEMBL26031834 0.78 NR4A2 (0.59) NR4A2ALOX5MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6495541-B1 POTENTIATION OF ANTICANCER THERAPIES AND INHIBITION OF NEUROTOXICITY CONSEQUENT TO STROKE, HEAD TRAUMA, AND NEURO-DEGENERATIVE DISEASES; SUCH AS 2-BROMO-3,4-DIHYDROPYRROLO-(4,3,2-DE)ISOGUINOLIN-5-ONE AGOURON PHARMACEUTICALS, INC. 2002-12-17 US disclosed