SCHEMBL7653574

SCHEMBL7653574

COc1ccc(Cn2c(=O)c3cc(CC(=O)O)ccc3n(C)c2=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
KDM4E B2RXH2 3/20 0.54
MAPT P10636 2/20 0.54
HPGD P15428 2/20 0.54
HSD17B10 Q99714 2/20 0.54
TSHR P16473 3/20 0.49
LMNA P02545 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
PMP22 Q01453 2/20 0.49
MMP13 P45452 1/20 0.49
SLC22A8 Q8TCC7 1/20 0.49
MEN1 O00255 1/20 0.49
RGS12 O14924 1/20 0.49
PKM P14618 1/20 0.49
NFKB1 P19838 1/20 0.49
MAPK1 P28482 1/20 0.49
GNAI1 P63096 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6256616 0.86 MMP13 (0.59) ALDH1A1MAPTLMNAMMP13SLC22A8
SCHEMBL6724632 0.85 MMP13 (0.53) ALDH1A1KDM4EMAPTLMNAMMP13
SCHEMBL10085642 0.83 TP53 (0.51) ALDH1A1KDM4ELMNAPARGTP53
SCHEMBL7634243 0.83 TP53 (0.57) MAPTMMP13SLC22A8PARGTP53
SCHEMBL5696996 0.81 MMP13 (0.55) LMNAMMP13SLC22A8KMT2APARG
SCHEMBL6234634 0.80 MMP13 (0.58) ALDH1A1KDM4EMAPTLMNAMMP13
SCHEMBL7018313 0.79 MMP13 (0.59) ALDH1A1MAPTLMNAMMP13SLC22A8
SCHEMBL6466889 0.79 P2RX4 (0.64) ALDH1A1KDM4EMAPTLMNAMEN1
SCHEMBL5922715 0.79 MMP13 (0.52) ALDH1A1KDM4EMAPTHSD17B10TSHR
SCHEMBL7100732 0.79 PIK3CD (0.51) ALDH1A1KDM4EMAPTLMNAMMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed