SCHEMBL7634243

SCHEMBL7634243

COC(=O)c1ccc2c(c1)c(=O)n(Cc1ccc(OC)cc1)c(=O)n2C

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.57
MAPT P10636 1/20 0.54
PARG Q86W56 4/20 0.52
HDAC1 Q13547 4/20 0.51
HDAC8 Q9BY41 2/20 0.51
HDAC6 Q9UBN7 2/20 0.51
MMP13 P45452 1/20 0.51
SLC22A8 Q8TCC7 1/20 0.51
HDAC11 Q96DB2 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6463989 0.90 MMP13 (0.55) TP53MAPTPARGHDAC1HDAC8
SCHEMBL27588029 0.90 PARG (0.52) TP53MAPTPARGHDAC1HDAC8
SCHEMBL6256616 0.90 MMP13 (0.59) TP53MAPTPARGHDAC1HDAC8
SCHEMBL27588009 0.89 PARG (0.54) TP53PARGHDAC1HDAC8HDAC6
SCHEMBL27588034 0.89 PARG (0.52) TP53MAPTPARGHDAC1HDAC8
SCHEMBL7103213 0.89 PARG (0.52) TP53PARGHDAC1HDAC8HDAC6
SCHEMBL27588021 0.89 PARG (0.54) TP53PARGHDAC1HDAC8HDAC6
SCHEMBL6245488 0.89 MMP13 (0.60) TP53MAPTPARGHDAC1HDAC8
SCHEMBL27588051 0.88 HDAC1 (0.53) TP53PARGHDAC1HDAC8HDAC6
SCHEMBL7105028 0.88 MMP13 (0.59) TP53MAPTPARGHDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020193377-A1 Quinazolines as MMP-13 inhibitors ANDRIANJARA CHARLES (FR) 2002-12-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020193377-A1 Quinazolines as MMP-13 inhibitors MMP13, MMP9, MMP3 TP53 4351/4885MAPT 4823/4885PARG 3624/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.