SCHEMBL7653663

SCHEMBL7653663

CC1CN(c2ccc(C(=O)NC(CC(=O)O)NS(=O)(=O)c3ccccc3)cc2)CCN1c1ncccn1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A7 Q99884 1/20 0.42
HSD11B1 P28845 7/20 0.40
ITGB3 P05106 3/20 0.40
ITGA2B P08514 3/20 0.40
ITGAV P06756 2/20 0.40
CASR P41180 4/20 0.39
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7652021 0.90 ITGB3 (0.41) ITGB3ITGA2BITGAVCASRNPC1
SCHEMBL7654428 0.87 ITGB3 (0.48) SLC6A7ITGB3ITGA2BITGAVNPC1
SCHEMBL7651967 0.85 ITGB3 (0.49) HSD11B1ITGB3ITGA2BITGAVCASR
SCHEMBL7653647 0.83 ITGB3 (0.61) ITGB3ITGA2BITGAV
SCHEMBL7649898 0.83 ITGB3 (0.61) ITGB3ITGA2BITGAV
SCHEMBL7651415 0.83 ITGB3 (0.61) ITGB3ITGA2BITGAV
SCHEMBL7464453 0.79 ITGB3 (0.54) ITGB3ITGA2BITGAVCASRLMNA
SCHEMBL27551456 0.79 ITGB3 (0.51) ITGB3ITGA2BITGAVCASR
SCHEMBL382764 0.79 ITGB3 (0.51) ITGB3ITGA2BITGAVCASR
SCHEMBL7658101 0.78 ITGB3 (0.48) ITGB3ITGA2BITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US claimed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP claimed
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US disclosed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP disclosed