SCHEMBL7653910

SCHEMBL7653910

C=CCOC(=O)CNCc1c([N+](=O)[O-])ccc(Cl)c1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.38
ALDH1A1 P00352 3/20 0.34
THRB P10828 1/20 0.33
MAPT P10636 2/20 0.33
PLA2G1B P04054 1/20 0.33
ATG4B Q9Y4P1 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
VCAM1 P19320 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NPC1 O15118 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LMNA P02545 1/20 0.31
BACE1 P56817 1/20 0.31
HCAR3 P49019 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL273112 0.85 LMNA (0.45) TDP1ALDH1A1THRBMAPTKDM4E
Hydrochloric Acid SCHEMBL273187 0.84 LMNA (0.44) TDP1ALDH1A1THRBMAPTKDM4E
SCHEMBL27919377 0.83 TDP1 (0.44) TDP1ALDH1A1THRBMAPTKDM4E
Hydrochloric Acid SCHEMBL5710125 0.82 TDP1 (0.43) TDP1ALDH1A1THRBMAPTKDM4E
SCHEMBL2476369 0.82 TDP1 (0.38) TDP1ALDH1A1THRBMAPTMEN1
SCHEMBL7162754 0.81 ALDH1A1 (0.38) ALDH1A1KDM4EMEN1KMT2AL3MBTL1
SCHEMBL2476365 0.79 TDP1 (0.40) TDP1ALDH1A1THRBMAPTKDM4E
SCHEMBL2720971 0.79 TDP1 (0.47) TDP1ALDH1A1MAPTKDM4EMEN1
Hydrochloric Acid SCHEMBL4432331 0.78 MAPT (0.49) TDP1ALDH1A1MAPTKDM4EMEN1
SCHEMBL278949 0.72 TDP1 (0.51) TDP1ALDH1A1THRBMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994114-B1 Process for the preparation of imidazoquinazolinone derivatives SHIRE US INC (US) 2002-12-04 EP disclosed
EP-0994114-A2 Process for the preparation of imidazoquinazolinone derivatives ROBERTS LABORATORIES INC. (US) 2000-04-19 EP disclosed
US-5801245-A Process for the preparation of ethyl-N-(2,3 dichloro-6-nitrobenzyl) glycine ROBERTS LABORATORIES INC. (US) 1998-09-01 US disclosed
EP-0778258-A2 Process for the preparation of ethyl-n-(2,3 dichloro-6-nitrobenzyl) glycine ROBERTS LABORATORIES INC. (US) 1997-06-11 EP disclosed