SCHEMBL7654067

SCHEMBL7654067

CCN(CCN1CCN(Cc2cccc3ccccc23)C1=C(C#N)C#N)C(=O)c1ccc(CN2CCCCC2)cc1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.60
OPRM1 P35372 5/20 0.39
OPRK1 P41145 4/20 0.39
NPFFR1 Q9GZQ6 3/20 0.39
NPFFR2 Q9Y5X5 3/20 0.39
OPRD1 P41143 5/20 0.38
MBTPS1 Q14703 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7654053 0.87 HRH3 (0.60) HRH3OPRM1OPRK1NPFFR1NPFFR2
SCHEMBL7659427 0.85 HRH3 (0.67) HRH3OPRM1OPRK1NPFFR1NPFFR2
SCHEMBL7665094 0.84 HRH3 (0.60) HRH3OPRM1OPRK1NPFFR1NPFFR2
SCHEMBL7655725 0.83 HRH3 (0.66) HRH3OPRM1OPRK1NPFFR1NPFFR2
SCHEMBL7659514 0.83 RAPGEF3 (0.46) HRH3OPRM1OPRD1
SCHEMBL7655220 0.83 HRH3 (0.39) HRH3OPRM1OPRD1
SCHEMBL7664398 0.81 HRH3 (0.56) HRH3OPRM1OPRK1NPFFR1NPFFR2
SCHEMBL7656388 0.81 HRH3 (0.65) HRH3OPRM1OPRK1NPFFR1NPFFR2
SCHEMBL7656593 0.80 HRH3 (0.55) HRH3OPRM1OPRK1NPFFR1NPFFR2
SCHEMBL7663692 0.79 HRH3 (0.67) HRH3NPFFR1NPFFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002085861-A1 IMIDAZOLIDINE COMPOUNDS AND THEIR USE AS CXCR3 ANTAGONISTS MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-10-31 WO disclosed
US-6469002-B1 COMPOUNDS WHICH MODULATE CHEMOKINE RECEPTOR ACTIVITY AND ARE USEFUL IN TREATMENT OF INFLAMMATORY DISEASES MILLENNIUM PHARMACEUTICALS, INC. 2002-10-22 US disclosed