SCHEMBL7654420

SCHEMBL7654420

O=c1[nH]c(=O)n(CCCN2CCC(OC(c3ccccc3)c3ccccc3)CC2)c2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.52
DRD2 P14416 3/20 0.52
HTR2A P28223 3/20 0.52
LMNA P02545 3/20 0.52
CHRM2 P08172 3/20 0.52
CHRM1 P11229 3/20 0.52
SLC6A2 P23975 3/20 0.52
ADRA1A P35348 3/20 0.52
DRD3 P35462 3/20 0.52
SLC6A3 Q01959 3/20 0.52
KCNH2 Q12809 3/20 0.52
MLNR O43193 2/20 0.52
NR1I2 O75469 2/20 0.52
ADORA3 P0DMS8 2/20 0.52
ADRA2C P18825 2/20 0.52
CHRM3 P20309 2/20 0.52
HTR2C P28335 2/20 0.52
SLC6A4 P31645 2/20 0.52
HRH1 P35367 2/20 0.52
OPRK1 P41145 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7649496 0.98 BCHE (0.53) P2RX7DRD2HTR2ALMNACHRM2
SCHEMBL7648364 0.97 P2RX7 (0.53) P2RX7DRD2HTR2ALMNACHRM2
SCHEMBL11205572 0.89 P2RX7 (0.66) P2RX7DRD2HTR2ALMNACHRM2
SCHEMBL7652682 0.88 BCHE (0.48) P2RX7DRD2HTR2ALMNACHRM2
SCHEMBL7656321 0.87 BCHE (0.48) P2RX7DRD2HTR2ALMNACHRM2
SCHEMBL7652277 0.87 BCHE (0.53) P2RX7DRD2HTR2ALMNASLC6A2
SCHEMBL7651720 0.87 BCHE (0.48) P2RX7DRD2HTR2ALMNACHRM2
SCHEMBL7654569 0.87 BCHE (0.53) P2RX7DRD2HTR2ALMNASLC6A2
SCHEMBL11369359 0.86 P2RX7 (0.66) P2RX7DRD2HTR2ALMNACHRM2
SCHEMBL7653211 0.85 BCHE (0.46) P2RX7DRD2HTR2ALMNACHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-11152275-A None JP disclosed
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed
JP-H11152275-A NITROGEN-CONTAINING CONDENSED RING COMPOUND, ITS PRODUCTION AND AGENT TAKEDA CHEM IND LTD 1999-06-08 JP disclosed