SCHEMBL7654569

SCHEMBL7654569

O=c1[nH]c(=O)n(CCCCN2CCC(OC(c3ccccc3)c3ccccc3)CC2)c2ccc(Cl)cc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 8/20 0.53
USP2 O75604 2/20 0.50
CYP1A2 P05177 2/20 0.50
CYP2D6 P10635 2/20 0.50
HTR1A P08908 2/20 0.50
MEN1 O00255 1/20 0.50
SLC22A2 O15244 1/20 0.50
NR1I2 O75469 1/20 0.50
GMNN O75496 1/20 0.50
LMNA P02545 1/20 0.50
GLA P06280 1/20 0.50
ADRB2 P07550 1/20 0.50
ADRB1 P08588 1/20 0.50
CYP3A4 P08684 1/20 0.50
ADRA2A P08913 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
DRD2 P14416 1/20 0.50
ADRA2B P18089 1/20 0.50
ADRA2C P18825 1/20 0.50
RXRA P19793 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7652277 0.93 BCHE (0.53) BCHEUSP2CYP1A2CYP2D6HTR1A
SCHEMBL7656321 0.89 BCHE (0.48) BCHECYP1A2CYP2D6HTR1AMEN1
SCHEMBL7651720 0.89 BCHE (0.48) BCHECYP1A2CYP2D6HTR1AMEN1
SCHEMBL7649496 0.89 BCHE (0.53) BCHECYP1A2CYP2D6HTR1AMEN1
SCHEMBL7648364 0.88 P2RX7 (0.53) BCHECYP1A2CYP2D6HTR1AMEN1
SCHEMBL7653124 0.88 BCHE (0.55) BCHECYP1A2CYP2D6HTR1AMEN1
SCHEMBL7659052 0.87 BCHE (0.46) BCHECYP1A2CYP2D6HTR1AMEN1
SCHEMBL7654420 0.87 P2RX7 (0.52) BCHECYP1A2CYP2D6HTR1AMEN1
SCHEMBL7652082 0.86 BCHE (0.56) BCHEHPGDSP2RX7
SCHEMBL7652273 0.86 BCHE (0.49) BCHECYP1A2CYP2D6HTR1AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed