SCHEMBL7654440

SCHEMBL7654440

O=Cc1ccccc1-c1ccc(Cn2cncn2)cc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 14/20 0.56
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
HTT P42858 1/20 0.41
STS P08842 2/20 0.41
XDH P47989 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6693307 0.79 CYP19A1 (0.61) CYP19A1HDAC1HDAC6SMN1; SMN2HTT
SCHEMBL7674570 0.78 CYP19A1 (0.79) CYP19A1HDAC1HDAC6SMN1; SMN2LMNA
SCHEMBL950133 0.78 CYP19A1 (0.62) CYP19A1HDAC1HDAC6SMN1; SMN2
SCHEMBL7657762 0.78 CYP19A1 (0.43) CYP19A1HDAC1HDAC6STS
SCHEMBL15688800 0.77 CYP19A1 (0.71) CYP19A1HDAC1HDAC6STS
SCHEMBL16494597 0.77 CYP19A1 (0.53) CYP19A1HDAC1HDAC6MAPT
SCHEMBL6700110 0.76 CYP19A1 (0.56) CYP19A1HDAC1HDAC6SMN1; SMN2HTT
SCHEMBL7655658 0.76 CYP19A1 (0.75) CYP19A1STS
SCHEMBL17159812 0.75 CYP19A1 (0.80) CYP19A1HDAC1HDAC6
SCHEMBL7653403 0.74 CYP19A1 (0.37) CYP19A1SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358984-B1 FOR THERAPY OF HYPERTENSION AND/OR DISEASES SUCH AS HEART AND RENAL DISEASES LEAD CHEMICAL CO., LTD. (JP) 2002-03-19 US disclosed
US-6232335-B1 A BIPHENYL TRIAZOLE COMPOUND USEFUL AS A ANGIOTENSIN II CONVERTING ENZYME INHIBITORS EFFECTIVE IN THE TREATMENT OF HYPERTENSION OR HEART FAILURE LEAD CHEMICAL CO., LTD. (JP) 2001-05-15 US disclosed