SCHEMBL7657762

SCHEMBL7657762

O=C1CC(=O)/C(=C/c2ccccc2-c2ccc(Cn3cncn3)cc2)N1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 15/20 0.43
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
STS P08842 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
FLT1 P17948 1/20 0.34
KDR P35968 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7657427 0.78 FLT3 (0.31)
SCHEMBL7654440 0.78 CYP19A1 (0.56) CYP19A1HDAC1HDAC6STS
SCHEMBL7654639 0.73 CYP19A1 (0.42) CYP19A1HDAC1HDAC6
SCHEMBL6693307 0.69 CYP19A1 (0.61) CYP19A1HDAC1HDAC6
SCHEMBL8300516 0.68 ACHE (0.31)
SCHEMBL7674570 0.68 CYP19A1 (0.79) CYP19A1HDAC1HDAC6STS
SCHEMBL15688800 0.67 CYP19A1 (0.71) CYP19A1HDAC1HDAC6STS
SCHEMBL8300436 0.66 ACHE (0.31)
SCHEMBL6700110 0.66 CYP19A1 (0.56) CYP19A1HDAC1HDAC6KDR
SCHEMBL7655658 0.66 CYP19A1 (0.75) CYP19A1STS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358984-B1 FOR THERAPY OF HYPERTENSION AND/OR DISEASES SUCH AS HEART AND RENAL DISEASES LEAD CHEMICAL CO., LTD. (JP) 2002-03-19 US disclosed
US-6232335-B1 A BIPHENYL TRIAZOLE COMPOUND USEFUL AS A ANGIOTENSIN II CONVERTING ENZYME INHIBITORS EFFECTIVE IN THE TREATMENT OF HYPERTENSION OR HEART FAILURE LEAD CHEMICAL CO., LTD. (JP) 2001-05-15 US disclosed