SCHEMBL7654816

SCHEMBL7654816

CCC(C(=O)O)n1c(=O)c2ccccc2n(CC)c1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.55
POLB P06746 2/20 0.50
KDM4E B2RXH2 10/20 0.49
ALDH1A1 P00352 6/20 0.49
MAPK8 P45983 1/20 0.48
RCE1 Q9Y256 1/20 0.48
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
HTT P42858 1/20 0.46
RECQL P46063 2/20 0.46
MAPT P10636 2/20 0.45
PKM P14618 1/20 0.45
MDM2 Q00987 1/20 0.45
TP53 P04637 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HDAC1 Q13547 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7648362 0.85 PGR (0.56) PGRPOLBKDM4EALDH1A1MAPK8
SCHEMBL10673575 0.82 MAPK8 (0.54) PGRPOLBKDM4EALDH1A1MAPK8
SCHEMBL7149835 0.78 POLB (0.64) POLBKDM4EALDH1A1HPGDRECQL
SCHEMBL3685766 0.78 CMA1 (0.70)
SCHEMBL3688506 0.78 CMA1 (0.70)
SCHEMBL3688933 0.78 CMA1 (0.70)
SCHEMBL4570289 0.77 CMA1 (0.51) POLB
SCHEMBL8472327 0.77 PGR (0.52) PGRKDM4EALDH1A1MAPK8RCE1
SCHEMBL8700032 0.76 MAPT (0.56) PGRPOLBKDM4EALDH1A1MAPK8
SCHEMBL3647510 0.75 CMA1 (0.79) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed