SCHEMBL7654930

SCHEMBL7654930

O=c1ccc(-c2c(-c3ccccc3)nn3ccccc23)nn1-c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.60
IGF1R P08069 2/20 0.52
MAPK1 P28482 5/20 0.46
MAPK14 Q16539 2/20 0.46
MAPK3 P27361 1/20 0.46
AKT1 P31749 1/20 0.44
EGFR P00533 2/20 0.43
RAF1 P04049 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43
GSK3B P49841 1/20 0.43
PDE5A O76074 1/20 0.38
PDE3A Q14432 1/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7664915 0.89 ADORA1 (0.53) ADORA1IGF1RMAPK1MAPK14MAPK3
SCHEMBL8809138 0.84 ADORA1 (0.64) ADORA1IGF1RMAPK1MAPK14MAPK3
SCHEMBL5798902 0.84 ADORA1 (0.55) ADORA1IGF1RMAPK1MAPK14MAPK3
SCHEMBL5798621 0.84 ADORA1 (0.55) ADORA1IGF1RMAPK1MAPK14MAPK3
SCHEMBL5795745 0.84 ADORA1 (0.55) ADORA1IGF1RMAPK1MAPK14MAPK3
SCHEMBL7658127 0.81 ADORA1 (0.53) ADORA1IGF1RMAPK1MAPK14MAPK3
SCHEMBL7039587 0.81 ADORA1 (0.57) ADORA1IGF1RMAPK1MAPK14MAPK3
SCHEMBL7299931 0.81 ADORA1 (0.57) ADORA1IGF1RMAPK1MAPK14MAPK3
SCHEMBL7304113 0.80 ADORA1 (0.68) ADORA1IGF1RMAPK1PDE3A
SCHEMBL7295203 0.79 ADORA1 (0.73) ADORA1IGF1RMAPK1MAPK14MAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355640-B1 TREATMENT OF HYPERTENSION, UROGENITAL DISORDERS AND FORMED BY WITTIG REACTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-03-12 US disclosed
US-5773530-A USEFUL AS PSYCHOSTIMULANTS, ANTIHYPERTENSIVE AGENTS AND REMEDIES FOR RENAL FAILURE, DIURETICS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-06-30 US disclosed