SCHEMBL765495

SCHEMBL765495

CC(O)C(O)(c1ccccc1)[C@H](C)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP1A2 P05177 1/20 0.38
KDM4E B2RXH2 1/20 0.38
PABPC1 P11940 1/20 0.38
APOBEC3A P31941 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
TSHR P16473 1/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
CHRM3 P20309 1/20 0.37
ALOX15 P16050 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
TTR P02766 1/20 0.35
GRIN1 Q05586 4/20 0.35
GRIN2A Q12879 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18096775 0.78 CYP2C19 (0.40) ALDH1A1CYP2D6CYP2C19HSD17B10CYP1A2
SCHEMBL27932553 0.77 ALDH1A1 (0.42) ALDH1A1CYP2D6CYP2C19HSD17B10CYP1A2
SCHEMBL9723670 0.77 CYP2D6 (0.48) ALDH1A1CYP2D6CYP2C19HSD17B10CYP1A2
SCHEMBL29150945 0.76 ALDH1A1 (0.39) ALDH1A1CYP2D6CYP2C19HSD17B10CYP1A2
SCHEMBL21963443 0.76 ALDH1A1 (0.39) ALDH1A1CYP2D6CYP2C19HSD17B10CYP1A2
SCHEMBL29150948 0.76 ALDH1A1 (0.39) ALDH1A1CYP2D6CYP2C19HSD17B10CYP1A2
SCHEMBL301345 0.74 ALDH1A1 (0.57) ALDH1A1CYP2D6CYP2C19HSD17B10CYP1A2
SCHEMBL6021075 0.74 ALDH1A1 (0.57) ALDH1A1CYP2D6CYP2C19HSD17B10CYP1A2
SCHEMBL7196262 0.72 ALDH1A1 (0.45) ALDH1A1CYP2D6CYP2C19HSD17B10CYP1A2
SCHEMBL27656872 0.72 ALDH1A1 (0.43) ALDH1A1CYP2D6CYP2C19HSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954668-B9 HOMO- AND HETEROCYCLIC COMPOUNDS SUITABLE AS CETP INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2012-03-21 EP disclosed
EP-1954668-B1 HOMO- AND HETEROCYCLIC COMPOUNDS SUITABLE AS CETP INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2011-09-28 EP disclosed