SCHEMBL7655419

SCHEMBL7655419

Cc1nc(Cl)cc(N2CCC(=O)CC2)n1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.41
KMT2A Q03164 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.37
PIM1 P11309 1/20 0.36
PIM2 Q9P1W9 1/20 0.36
USP2 O75604 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SORD Q00796 2/20 0.34
CHRM4 P08173 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3406103 0.82 KMT2A (0.54) KMT2ACYP1A2CYP2D6MAPTUSP2
SCHEMBL3413188 0.81 KMT2A (0.53) KMT2ACYP1A2CYP2D6MAPTUSP2
SCHEMBL17893818 0.79 PIM1 (0.40) KMT2ACYP1A2CYP2D6MAPTLMNA
SCHEMBL15956636 0.79 HTR3A (0.53) KMT2AHRH4HTR3EHTR3BHTR3A
SCHEMBL30353341 0.78 CYP1A2 (0.66) KMT2ACYP1A2CYP2D6MAPTPOLB
SCHEMBL20905447 0.78 KMT2A (0.51) KMT2ACYP1A2CYP2D6MAPTCHRM4
SCHEMBL913131 0.78 CYP1A2 (0.66) KMT2ACYP1A2CYP2D6MAPTPOLB
Hydrochloric Acid SCHEMBL1854981 0.77 KMT2A (0.50) KMT2ACYP1A2CYP2D6MAPTCHRM4
SCHEMBL11963431 0.76 GBA1 (0.42) KMT2ACYP1A2CYP2D6MAPTLMNA
SCHEMBL5429458 0.75 LMNA (0.46) CYP17A1KMT2ACYP1A2CYP2D6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6335341-B1 ANTICHOLESTEROL AGENTS; ATHEROSCLEROSIS ZENECA LIMITED (GB) 2002-01-01 US disclosed
EP-1000057-A1 PYRIDYL- AND PYRIMIDYL-HETEROCYCLIC COMPOUNDS INHIBITING OXIDO SQUALENE-CYCLASE AstraZeneca UK Limited (GB) 2000-05-17 EP disclosed
WO-1999006395-A1 PYRIDYL- AND PYRIMIDYL-HETEROCYCLIC COMPOUNDS INHIBITING OXIDO SQUALENE-CYCLASE ZENECA LIMITED (GB) 1999-02-11 WO disclosed