SCHEMBL7655652

SCHEMBL7655652

CCc1ccccc1N(C)C(=O)Cn1c(=O)[nH]c2ccccc2c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.54
MPO P05164 3/20 0.49
ALDH1A1 P00352 4/20 0.49
KDM4E B2RXH2 3/20 0.49
HPGD P15428 3/20 0.49
NPEPPS P55786 1/20 0.49
MAPT P10636 2/20 0.48
LMNA P02545 1/20 0.48
HSD17B10 Q99714 2/20 0.47
MAPK1 P28482 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.42
GAA P10253 1/20 0.42
HAVCR2 Q8TDQ0 1/20 0.42
TSHR P16473 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA2B P29275 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11985495 0.78 CYP1A2 (0.67) CYP1A2MPOALDH1A1KDM4EHPGD
SCHEMBL13332558 0.75 CYP1A2 (0.62) CYP1A2ALDH1A1KDM4EHPGDMAPT
SCHEMBL3311524 0.74 ALDH1A1 (0.73) CYP1A2MPOALDH1A1KDM4EHPGD
SCHEMBL3312291 0.72 CYP1A2 (0.61) CYP1A2MPOALDH1A1KDM4EHPGD
SCHEMBL32680072 0.72 CYP1A2 (0.61) CYP1A2MPOALDH1A1KDM4EHPGD
SCHEMBL9523849 0.72 CYP1A2 (1.00) CYP1A2MPOALDH1A1KDM4EHPGD
SCHEMBL10085092 0.72 POLB (0.43) CYP1A2ALDH1A1KDM4EMAPTLMNA
SCHEMBL7654823 0.71 MAPT (0.52) ALDH1A1KDM4EMAPTLMNAMAPK1
SCHEMBL8692730 0.70 CYP1A2 (0.76) CYP1A2MPOALDH1A1KDM4EHPGD
SCHEMBL3311829 0.69 CYP1A2 (0.57) CYP1A2MPOALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed