SCHEMBL7656239

SCHEMBL7656239

CN1Cc2cc(N)ccc2CC1(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.35
MAPT P10636 5/20 0.34
KDM4E B2RXH2 4/20 0.34
ALDH1A1 P00352 3/20 0.34
LMNA P02545 2/20 0.34
RAB9A P51151 2/20 0.34
HPGD P15428 2/20 0.34
NPC1 O15118 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PRKCI P41743 1/20 0.34
HSD17B3 P37058 1/20 0.34
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
PDK2 Q15119 1/20 0.33
RAD52 P43351 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29516233 0.79 BRD4 (0.42) MAPTSMN1; SMN2HSD17B3MEN1KMT2A
SCHEMBL1950822 0.76 MAPT (0.35) NR1H2MAPTKDM4EALDH1A1LMNA
SCHEMBL8028903 0.75 MAOA (0.43) ALDH1A1LMNAHPGDSMN1; SMN2OPRM1
SCHEMBL29516144 0.75 MAOA (0.43) ALDH1A1LMNAHPGDSMN1; SMN2OPRM1
SCHEMBL1950736 0.74 KDM4E (0.35) MAPTKDM4EALDH1A1LMNARAB9A
SCHEMBL188773 0.72 KDM4E (0.43) NR1H2MAPTKDM4EALDH1A1LMNA
SCHEMBL19927603 0.72 MAPT (0.41) MAPTKDM4EALDH1A1LMNARAB9A
SCHEMBL7652770 0.71 NR1H2 (0.40) NR1H2MAPTLMNARAB9AHSD17B3
Hydrochloric Acid SCHEMBL3572065 0.71 MAPT (0.46) NR1H2MAPTKDM4EALDH1A1LMNA
Hydrochloric Acid SCHEMBL30065224 0.71 MAPT (0.46) NR1H2MAPTKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023281417-A1 PYRIMIDINE COMPOUNDS FOR USE AS MAP4K1 INHIBITORS GLENMARK SPECIALTY S.A. (CH) 2023-01-12 WO disclosed
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed
EP-1104404-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 2001-06-06 EP disclosed
WO-2000009486-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSIVANTS SMITHKLINE BEECHAM P.L.C. (GB) 2000-02-24 WO disclosed
WO-2000007993-A1 SUBSTITUTED ISOQUINOLEINES AND THEIR USE AS ANTICONVULSIVANTS SMITHKLINE BEECHAM PLC (GB) 2000-02-17 WO disclosed