SCHEMBL7656918

SCHEMBL7656918

N#Cc1ccc(CO)cc1OC(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.51
KCNH2 Q12809 2/20 0.46
KCNJ1 P48048 1/20 0.46
MBOAT4 Q96T53 1/20 0.38
IDH1 O75874 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
S1PR1 P21453 2/20 0.37
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
RXRG P48443 1/20 0.37
ACACB O00763 1/20 0.37
FFAR1 O14842 2/20 0.36
FFAR4 Q5NUL3 1/20 0.36
SLC22A12 Q96S37 2/20 0.36
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
TMEM97 Q5BJF2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1918756 0.90 AR (0.51) ARKCNH2KCNJ1MBOAT4CYP11B1
SCHEMBL15210068 0.88 KCNH2 (0.50) ARKCNH2KCNJ1MBOAT4IDH1
SCHEMBL23791163 0.84 KCNJ1 (0.46) ARKCNH2KCNJ1MBOAT4IDH1
SCHEMBL2723153 0.82 RXRA (0.54) KCNH2KCNJ1S1PR1RXRARXRB
SCHEMBL2723065 0.81 KCNJ1 (0.47) ARKCNH2KCNJ1MBOAT4IDH1
SCHEMBL8157355 0.81 AR (0.52) ARCYP11B1CYP11B2S1PR1RXRA
SCHEMBL16822097 0.81 KCNH2 (0.50) ARKCNH2KCNJ1MBOAT4IDH1
SCHEMBL16961827 0.79 CYP4F2 (0.42) ARKCNH2RXRARXRBRXRG
SCHEMBL22954039 0.79 KCNH2 (0.48) ARKCNH2KCNJ1MBOAT4IDH1
SCHEMBL8709726 0.78 MBOAT4 (0.43) ARKCNH2KCNJ1MBOAT4S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900645-A1 3-PHENYLISOXAZOLIN DERIVATIVES WITH HERBICIDAL ACTION Bayer CropScience AG (DE) 2015-08-05 EP disclosed
US-6387903-B1 ANTICANCER AGENT; CARDIOVASCULAR DISORDERS; VIRICIDES MERCK & CO., INC. 2002-05-14 US disclosed
EP-1014984-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2000-07-05 EP disclosed
WO-1999009985-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1999-03-04 WO disclosed