SCHEMBL7657286

SCHEMBL7657286

Cc1ccc(C2(c3ccc(C)cc3)NC(=O)N(CCCN3CCC4(CC3)OC(=O)N(C)c3ccccc34)C2=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 1/20 0.51
HRH3 Q9Y5N1 1/20 0.51
SIGMAR1 Q99720 8/20 0.48
ADRA1A P35348 3/20 0.47
CNR1 P21554 1/20 0.43
ADRA1D P25100 2/20 0.42
ADRA1B P35368 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656122 0.88 HRH1 (0.43) HRH1HRH3SIGMAR1ADRA1ACNR1
SCHEMBL7660411 0.85 HRH1 (0.53) HRH1HRH3SIGMAR1ADRA1ACNR1
SCHEMBL7652320 0.85 HRH1 (0.54) HRH1HRH3SIGMAR1ADRA1AADRA1D
SCHEMBL7656937 0.83 HRH1 (0.45) HRH1HRH3SIGMAR1CNR1
SCHEMBL7681283 0.80 HRH1 (0.57) HRH1HRH3SIGMAR1ADRA1ACNR1
SCHEMBL7675906 0.79 HRH1 (0.54) HRH1HRH3SIGMAR1ADRA1ACNR1
SCHEMBL7653823 0.79 HRH1 (0.56) HRH1HRH3SIGMAR1ADRA1AADRA1D
Hydrochloric Acid SCHEMBL7664647 0.78 HRH1 (0.55) HRH1HRH3SIGMAR1ADRA1AADRA1D
SCHEMBL7652519 0.77 ADRA1A (0.40) HRH1HRH3SIGMAR1ADRA1ACNR1
SCHEMBL11718665 0.77 HRH1 (0.65) HRH1HRH3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436962-B1 ALPHA 1A ADRENERGIC RECEPTOR ANTAGONISTS; RELIEF FROM BENIGN PROSTATIC HYPERPLASIA BY LESS HINDERED URINE FLOW BY RELAXING SMOOTH MUSCLE TISSUE; WITH A TESTOSTERONE 5-ALPHA REDUCTASE INHIBITOR, FINASTERIDE; ACUTE AND CHRONIC RELIEF MERCK & CO., INC. 2002-08-20 US disclosed