SCHEMBL7657939

SCHEMBL7657939

CSC(C)C[C@H](NC(=O)c1ccc(NC(Cn2ccnc2)c2ccc(F)cc2)cc1Cc1ccc(F)cc1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
FNTA P49354 3/20 0.41
FNTB P49356 3/20 0.41
PGGT1B P53609 1/20 0.40
PTGS2 P35354 1/20 0.39
CYP51A1 Q16850 5/20 0.38
AGTR2 P50052 1/20 0.35
POLB P06746 1/20 0.35
CYP26A1 O43174 1/20 0.34
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7660347 0.89 FNTA (0.54) FNTAFNTB
SCHEMBL7656236 0.88 FNTA (0.49) CYP3A4CYP2C19CYP2D6CYP2C9FNTA
SCHEMBL7667477 0.87 FNTA (0.53) CYP3A4CYP2C19CYP2D6CYP2C9FNTA
SCHEMBL7665403 0.83 CYP19A1 (0.41) PTGS2CYP51A1POLB
SCHEMBL7657934 0.83 FNTA (0.46) CYP3A4CYP2C19CYP2D6CYP2C9FNTA
SCHEMBL7656299 0.82 FNTA (0.52) FNTAFNTB
SCHEMBL7657941 0.79 FNTA (0.37) CYP3A4CYP2C19CYP2D6CYP2C9FNTA
SCHEMBL7660599 0.78 FNTA (0.46) CYP3A4CYP2C19CYP2D6CYP2C9FNTA
SCHEMBL7668699 0.77 FNTA (0.51) FNTAFNTBPGGT1B
SCHEMBL7662078 0.76 FNTA (0.49) CYP3A4CYP2C19CYP2D6CYP2C9FNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6410539-B1 ANTICARCINOGENIC AGENTS ASTRAZENCA UK LIMITED (GB) 2002-06-25 US claimed