SCHEMBL7665403

SCHEMBL7665403

O=C(O)c1ccc(NC(Cn2ccnc2)c2ccc(F)cc2)cc1Cc1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.41
CYP51A1 Q16850 4/20 0.41
AURKA O14965 1/20 0.41
PDPK1 O15530 1/20 0.41
RPS6KB1 P23443 1/20 0.41
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
PTGS2 P35354 1/20 0.40
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656582 0.84 CYP51A1 (0.49) CYP19A1CYP51A1AURKAPDPK1RPS6KB1
SCHEMBL7660347 0.83 FNTA (0.54)
SCHEMBL7657939 0.83 CYP3A4 (0.41) CYP51A1PTGS2POLB
SCHEMBL7664949 0.83 PTGS2 (0.40) CYP19A1CYP51A1CYP11B1CYP11B2PTGS2
SCHEMBL7657941 0.81 FNTA (0.37) CYP19A1CYP51A1AURKAPDPK1RPS6KB1
SCHEMBL7657934 0.80 FNTA (0.46) CYP51A1PTGS2
SCHEMBL7656299 0.78 FNTA (0.52)
SCHEMBL8185720 0.78 CYP24A1 (0.52) CYP19A1
SCHEMBL7653706 0.76 PTGS2 (0.47) CYP51A1PTGS2
SCHEMBL7667709 0.76 PTGS2 (0.39) CYP19A1CYP51A1CYP11B1CYP11B2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6410539-B1 ANTICARCINOGENIC AGENTS ASTRAZENCA UK LIMITED (GB) 2002-06-25 US disclosed