SCHEMBL7659848

SCHEMBL7659848

COCCN1Cc2cc(NC(=O)c3ccc(C(C)C)c(C#N)c3)ccc2C(C)(C)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 7/20 0.39
DDR1 Q08345 4/20 0.37
DDR2 Q16832 4/20 0.37
L3MBTL3 Q96JM7 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
HSD17B10 Q99714 2/20 0.36
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
GAA P10253 1/20 0.36
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36
FPR1 P21462 1/20 0.36
FPR2 P25090 1/20 0.36
MEN1 O00255 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7993332 0.90 ROCK2 (0.45) ROCK2DDR1DDR2CYP3A4ALDH1A1
SCHEMBL7655182 0.89 ROCK2 (0.42) ROCK2CYP3A4
SCHEMBL7660384 0.80 ROCK2 (0.51) ROCK2CYP3A4ALDH1A1MAPTHSD17B10
SCHEMBL7660601 0.80 MAPT (0.44) ROCK2L3MBTL3CYP3A4ALDH1A1MAPT
SCHEMBL7662103 0.79 MAPT (0.45) ROCK2CYP3A4MAPTHSD17B10ALOX15
SCHEMBL7655775 0.79 ROCK2 (0.46) ROCK2CYP3A4ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL7653098 0.79 MAPT (0.43) ROCK2L3MBTL3CYP3A4ALDH1A1MAPT
SCHEMBL7659472 0.79 ROCK2 (0.43) ROCK2CYP3A4ALDH1A1MAPTHSD17B10
SCHEMBL7654987 0.79 ROCK2 (0.43) ROCK2DDR1DDR2L3MBTL3CYP3A4
SCHEMBL6295077 0.78 ROCK2 (0.58) ROCK2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed