SCHEMBL7659472

SCHEMBL7659472

CC(C)c1ccc(C(=O)Nc2ccc3c(c2)C(C)(C)N(C)CC3)cc1C#N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 11/20 0.43
GAA P10253 2/20 0.38
GFER P55789 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP26A1 O43174 1/20 0.38
PGR P06401 1/20 0.38
CYP3A4 P08684 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
RARA P10276 1/20 0.38
RARB P10826 1/20 0.38
RARG P13631 1/20 0.38
TBXA2R P21731 1/20 0.38
BLVRB P30043 1/20 0.38
MAPT P10636 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7653964 0.88 GAA (0.39) ROCK2GAAMEN1KMT2AMAPT
Hydrochloric Acid SCHEMBL7661203 0.87 GAA (0.39) ROCK2GAAMEN1KMT2AMAPT
SCHEMBL7662414 0.87 ROCK2 (0.37) ROCK2GAAMAPTSMN1; SMN2HTT
SCHEMBL6295077 0.84 ROCK2 (0.58) ROCK2CYP3A4
Hydrochloric Acid SCHEMBL6299497 0.83 ROCK2 (0.57) ROCK2CYP3A4
SCHEMBL7993332 0.83 ROCK2 (0.45) ROCK2MEN1KMT2ACYP26A1PGR
SCHEMBL7656532 0.81 ROCK2 (0.43) ROCK2
SCHEMBL7659848 0.79 ROCK2 (0.39) ROCK2GAAMEN1KMT2ACYP3A4
SCHEMBL7656812 0.78 CYP26A1 (0.38) ROCK2GAAMEN1KMT2ACYP26A1
SCHEMBL7654464 0.78 ROCK2 (0.41) ROCK2MEN1KMT2AMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed