SCHEMBL7662993

SCHEMBL7662993

COC(=O)c1ccc(N)cc1-c1ccc(F)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 4/20 0.63
SLC6A4 P31645 3/20 0.63
GAA P10253 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.50
NPC1 O15118 1/20 0.50
CASP3 P42574 1/20 0.50
RAB9A P51151 1/20 0.50
SENP8 Q96LD8 1/20 0.50
SENP7 Q9BQF6 1/20 0.50
SENP6 Q9GZR1 1/20 0.50
IKBKB O14920 1/20 0.49
LMNA P02545 1/20 0.48
PTGS1 P23219 2/20 0.45
KDM4E B2RXH2 3/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C19 P33261 2/20 0.44
PTGS2 P35354 1/20 0.44
CYP2C9 P11712 1/20 0.44
ALDH1A1 P00352 5/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31676847 0.87 SLC6A3 (0.71) SLC6A3SLC6A4SMN1; SMN2NPC1CASP3
SCHEMBL23354126 0.87 SLC6A3 (0.71) SLC6A3SLC6A4SMN1; SMN2NPC1CASP3
SCHEMBL2723555 0.85 SLC6A3 (0.63) SLC6A3SLC6A4GAASMN1; SMN2NPC1
SCHEMBL630047 0.84 GAA (0.58) SLC6A3SLC6A4GAASMN1; SMN2LMNA
SCHEMBL29775249 0.84 GAA (0.58) SLC6A3SLC6A4GAASMN1; SMN2LMNA
Hydrochloric Acid SCHEMBL6625663 0.83 GAA (0.57) SLC6A3SLC6A4GAASMN1; SMN2LMNA
SCHEMBL7563000 0.83 SLC6A3 (0.65) SLC6A3SLC6A4GAASMN1; SMN2NPC1
SCHEMBL7249446 0.83 SLC6A3 (0.65) SLC6A3SLC6A4SMN1; SMN2NPC1CASP3
SCHEMBL6783755 0.82 KDM4E (0.63) SLC6A3SLC6A4SMN1; SMN2NPC1CASP3
SCHEMBL16741757 0.81 IKBKB (0.51) IKBKBPTGS1CYP1A2CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6410539-B1 ANTICARCINOGENIC AGENTS ASTRAZENCA UK LIMITED (GB) 2002-06-25 US disclosed
EP-1054865-A1 FARNESYL TRANSFERASE INHIBITORS AstraZeneca UK Limited (GB) 2000-11-29 EP disclosed
EP-1025089-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS FARNESYL PROTEIN TRANSFERASE INHIBITORS ZENECA LIMITED (GB) 2000-08-09 EP disclosed
WO-1999041235-A1 FARNESYL TRANSFERASE INHIBITORS ASTRAZENECA UK LIMITED (GB) 1999-08-19 WO disclosed
WO-1999020612-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS FARNESYL PROTEIN TRANSFERASE INHIBITORS ASTRAZENECA UK LIMITED (GB) 1999-04-29 WO disclosed