SCHEMBL7664685

SCHEMBL7664685

CC(/C=C/C(F)=C(/C)c1ccc2c(c1)N(C(C)C)CCN2C(C)C)=C\C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RXRA P19793 11/20 0.38
RXRB P28702 7/20 0.38
RXRG P48443 6/20 0.38
RARA P10276 11/20 0.38
RARB P10826 11/20 0.38
PPARG P37231 4/20 0.38
RARG P13631 7/20 0.34
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
PKM P14618 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7664689 1.00 RXRA (0.38) RXRARXRBRXRGRARARARB
SCHEMBL7674374 0.86 RXRA (0.36) RXRARXRBRXRGRARARARB
SCHEMBL7667037 0.86 HDAC1 (0.38) RXRARXRBRXRGRARARARB
SCHEMBL7667028 0.86 HDAC1 (0.38) RXRARXRBRXRGRARARARB
SCHEMBL7667039 0.86 HDAC1 (0.38) RXRARXRBRXRGRARARARB
SCHEMBL7674365 0.86 RXRA (0.36) RXRARXRBRXRGRARARARB
SCHEMBL7664500 0.85 HDAC1 (0.36) RXRARXRBRXRGRARARARB
SCHEMBL7669724 0.85 RXRA (0.37) RXRARXRBRXRGRARARARB
SCHEMBL7664742 0.85 HDAC1 (0.36) RXRARXRBRXRGRARARARB
SCHEMBL7669731 0.85 RXRA (0.37) RXRARXRBRXRGRARARARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420363-B1 Mono- or polyenic carboxylic acid derivatives EISAI CO., LTD. (JP) 2002-07-16 US disclosed
US-6291508-B1 POTENT ABILITY TO BIND TO RETINOIC ACID RECEPTORS THUS USEFUL IN TREATING PSORIASIS AND RHEUMATOID ARTHRITIS. EISAI CO., LTD. (JP) 2001-09-18 US disclosed
US-6133283-A Mono- or polyenic carboxylic acid derivatives EISAI CO., LTD. (JP) 2000-10-17 US disclosed
US-6030964-A BINDS TO RETINOIC ACID RECEPTORS AND USEFUL FOR TREATING PSORIASIS, AUTOIMMUNE DISEASES, TUMORS, RHEUMATOID ARTHRITIS AND FOR INDUCING IMMUNOSUPPRESSION IN ORGAN TRANSPLANTATION EISAI CO., LTD. (JP) 2000-02-29 US disclosed
US-5977125-A Mono-or polyenic carboxylic acid derivatives EISAI CO., LTD. (JP) 1999-11-02 US disclosed
EP-0790228-A1 MONO- OR POLYENIC CARBOXYLIC ACID DERIVATIVE Eisai Co., Ltd. (JP) 1997-08-20 EP disclosed