SCHEMBL7674374

SCHEMBL7674374

CC(C=CC(F)=C(C)c1ccc2c(c1)N(C(C)C)CCC2)=CC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RXRA P19793 11/20 0.36
RARA P10276 7/20 0.36
RARB P10826 7/20 0.36
RXRB P28702 6/20 0.36
RXRG P48443 6/20 0.36
PPARG P37231 4/20 0.36
RARG P13631 3/20 0.33
LMNA P02545 2/20 0.33
TP53 P04637 1/20 0.33
HDAC1 Q13547 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
PMP22 Q01453 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GFER P55789 1/20 0.32
MEN1 O00255 1/20 0.32
TSHR P16473 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7674365 1.00 RXRA (0.36) RXRARARARARBRXRBRXRG
SCHEMBL7667028 0.92 HDAC1 (0.38) RXRARARARARBRXRBRXRG
SCHEMBL7667037 0.92 HDAC1 (0.38) RXRARARARARBRXRBRXRG
SCHEMBL7667039 0.92 HDAC1 (0.38) RXRARARARARBRXRBRXRG
SCHEMBL7664742 0.89 HDAC1 (0.36) RXRARARARARBRXRBRXRG
SCHEMBL7664500 0.89 HDAC1 (0.36) RXRARARARARBRXRBRXRG
SCHEMBL7664506 0.89 HDAC1 (0.36) RXRARARARARBRXRBRXRG
SCHEMBL7667613 0.88 KDM4E (0.36) RXRARARARARBRXRBRXRG
SCHEMBL7667605 0.88 KDM4E (0.36) RXRARARARARBRXRBRXRG
SCHEMBL7664685 0.86 RXRA (0.38) RXRARARARARBRXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420363-B1 Mono- or polyenic carboxylic acid derivatives EISAI CO., LTD. (JP) 2002-07-16 US disclosed
US-6291508-B1 POTENT ABILITY TO BIND TO RETINOIC ACID RECEPTORS THUS USEFUL IN TREATING PSORIASIS AND RHEUMATOID ARTHRITIS. EISAI CO., LTD. (JP) 2001-09-18 US disclosed
US-6133283-A Mono- or polyenic carboxylic acid derivatives EISAI CO., LTD. (JP) 2000-10-17 US disclosed
US-6030964-A BINDS TO RETINOIC ACID RECEPTORS AND USEFUL FOR TREATING PSORIASIS, AUTOIMMUNE DISEASES, TUMORS, RHEUMATOID ARTHRITIS AND FOR INDUCING IMMUNOSUPPRESSION IN ORGAN TRANSPLANTATION EISAI CO., LTD. (JP) 2000-02-29 US disclosed
US-5977125-A Mono-or polyenic carboxylic acid derivatives EISAI CO., LTD. (JP) 1999-11-02 US disclosed
EP-0790228-A1 MONO- OR POLYENIC CARBOXYLIC ACID DERIVATIVE Eisai Co., Ltd. (JP) 1997-08-20 EP disclosed