SCHEMBL7665490

SCHEMBL7665490

CC(=O)On1ncc2cc3[nH]c(=O)c(-c4cn(Cc5cccc(CN)n5)c5ccccc45)nc3cc21

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 1/20 0.33
CA12 O43570 3/20 0.31
CA1 P00915 3/20 0.31
CA9 Q16790 3/20 0.31
CA2 P00918 2/20 0.31
KDR P35968 1/20 0.31
CHRM1 P11229 1/20 0.31
SAE1 Q9UBE0 1/20 0.30
UBA2 Q9UBT2 1/20 0.30
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7662876 0.91 CA12 (0.37) CA12CA1CA9CA2KDR
SCHEMBL7659554 0.90 CA12 (0.36) CA12CA1CA9CA2KDR
SCHEMBL7657220 0.86 CAMK2D (0.42) KDR
SCHEMBL7652600 0.85 ACKR3 (0.33) ACKR3CA12CA1CA9CA2
Acetic Acid SCHEMBL7662873 0.85 CA12 (0.37) ACKR3CA12CA1CA9CA2
SCHEMBL12856392 0.83 MEN1 (0.40) ACKR3CA12CA1CA9CA2
Acetic Acid SCHEMBL7665482 0.82 CA12 (0.36) ACKR3CA12CA1CA9CA2
Acetic Acid SCHEMBL7852409 0.82 CA12 (0.36) ACKR3CA12CA1CA9CA2
Acetic Acid SCHEMBL8516673 0.81 CAMK2D (0.37) ACKR3CA12CA1CA9CA2
Acetic Acid SCHEMBL7658062 0.81 ACKR3 (0.35) ACKR3CA12CA1CA9CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6458792-B1 MEDICAMENT FOR THE TREATMENT OF INFLAMMATORY, IMMUNOLOGICAL, BRONCHOPULMONARY, CARDIOVASCULAR, ONCOLOGICAL OR CNS-DEGENERATIVE DISORDERS. ASTRAZENECA AB (SE) 2002-10-01 US disclosed
EP-1071683-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2001-01-31 EP disclosed
WO-1999046264-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 1999-09-16 WO disclosed