SCHEMBL7667240

SCHEMBL7667240

Cc1cc(N2CCC(NC(=O)OC(C)(C)C)C2)ccc1NC(=O)CC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.47
HSD11B1 P28845 2/20 0.43
SUV39H2 Q9H5I1 6/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
KMT2A Q03164 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
EPHX1 P07099 1/20 0.40
EPHX2 P34913 1/20 0.40
PIM1 P11309 1/20 0.40
PIM3 Q86V86 1/20 0.40
PIM2 Q9P1W9 1/20 0.40
ABCB11 O95342 1/20 0.40
HRH3 Q9Y5N1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7660361 0.81 EPHX2 (0.54) P2RX7MEN1ALDH1A1KMT2ANPSR1
SCHEMBL7607645 0.81 HRH3 (0.43) SUV39H2PIM1PIM3PIM2HRH3
SCHEMBL7242505 0.76 SUV39H2 (0.50) SUV39H2PIM1PIM3PIM2
SCHEMBL6486070 0.76 SUV39H2 (0.50) SUV39H2PIM1PIM3PIM2
SCHEMBL25453975 0.75 SUV39H2 (0.55) SUV39H2PIM1PIM3PIM2
SCHEMBL1350982 0.74 SUV39H2 (0.48) SUV39H2PIM1PIM3PIM2
SCHEMBL1350984 0.74 SUV39H2 (0.48) SUV39H2PIM1PIM3PIM2
SCHEMBL7235725 0.74 SUV39H2 (0.48) SUV39H2PIM1PIM3PIM2
SCHEMBL4508024 0.73 P2RX7 (0.50) P2RX7EPHX1
SCHEMBL30371860 0.73 RAD52 (0.58) MEN1ALDH1A1KMT2ANPSR1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492355-B1 Adamantane derivatives ASTRAZENECA AB (SE) 2002-12-10 US disclosed