SCHEMBL7667449

SCHEMBL7667449

CC(C=CC=C(C)c1ccc2c(ccn2C(C)C)c1)=CC(=O)O

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RARG P13631 8/20 0.49
RXRA P19793 8/20 0.49
RARA P10276 5/20 0.49
RARB P10826 5/20 0.49
RXRB P28702 1/20 0.47
RXRG P48443 1/20 0.47
PPARG P37231 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7667442 1.00 RARG (0.49) RARGRXRARARARARBRXRB
SCHEMBL7664518 0.85
SCHEMBL7664512 0.85
SCHEMBL7667024 0.81 PPARG (0.38) RXRARARARARBRXRBRXRG
SCHEMBL9465521 0.76
SCHEMBL9465508 0.76
SCHEMBL10562459 0.75 RXRA (0.57) RARGRXRARARARARBRXRB
SCHEMBL10558322 0.74 RXRA (0.54) RARGRXRARARARARBRXRB
SCHEMBL4740640 0.74 HCAR3 (0.55) RXRAPPARG
SCHEMBL9033451 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420363-B1 Mono- or polyenic carboxylic acid derivatives EISAI CO., LTD. (JP) 2002-07-16 US disclosed
US-6133283-A Mono- or polyenic carboxylic acid derivatives EISAI CO., LTD. (JP) 2000-10-17 US disclosed
US-6030964-A BINDS TO RETINOIC ACID RECEPTORS AND USEFUL FOR TREATING PSORIASIS, AUTOIMMUNE DISEASES, TUMORS, RHEUMATOID ARTHRITIS AND FOR INDUCING IMMUNOSUPPRESSION IN ORGAN TRANSPLANTATION EISAI CO., LTD. (JP) 2000-02-29 US disclosed
US-5977125-A Mono-or polyenic carboxylic acid derivatives EISAI CO., LTD. (JP) 1999-11-02 US disclosed
EP-0790228-A1 MONO- OR POLYENIC CARBOXYLIC ACID DERIVATIVE Eisai Co., Ltd. (JP) 1997-08-20 EP disclosed