SCHEMBL7667643

SCHEMBL7667643

COc1cccc(-c2nc(=O)c3cc(N(C)C)ccc3[nH]2)c1

nearest known ligand 0.69

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.54
CYP1A2 P05177 1/20 0.54
VDR P11473 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2B6 P20813 1/20 0.54
AHR P35869 1/20 0.54
NR1I3 Q14994 1/20 0.54
AURKA O14965 2/20 0.49
PARP1 P09874 1/20 0.47
MEN1 O00255 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
KMT2A Q03164 1/20 0.47
PIN1 Q13526 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7674412 0.88 NR1I2 (0.61) NR1I2CYP1A2VDRCYP2C9CYP2B6
SCHEMBL7668642 0.83 LMNA (0.56) NR1I2CYP1A2VDRCYP2C9CYP2B6
SCHEMBL7665249 0.83 NR1I2 (0.56) NR1I2CYP1A2VDRCYP2C9CYP2B6
SCHEMBL7668615 0.83 NR1I2 (0.72) NR1I2CYP1A2VDRCYP2C9CYP2B6
SCHEMBL7671162 0.81 NR1I2 (0.55) NR1I2CYP1A2VDRCYP2C9CYP2B6
SCHEMBL31238239 0.79 HPGD (0.70) MEN1MAPTHPGDKMT2A
SCHEMBL8980334 0.79 HPGD (0.70) MEN1MAPTHPGDKMT2A
SCHEMBL7669056 0.78 TUBB4A (0.67) NR1I2CYP1A2VDRCYP2C9CYP2B6
SCHEMBL7675227 0.77 TUBB4A (0.66) NR1I2CYP1A2VDRCYP2C9CYP2B6
SCHEMBL7675597 0.76 MAPT (0.50) NR1I2CYP1A2VDRCYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6479499-B1 INHIBITORS OF TUBULIN POLYMERIZATION NATIONAL SCIENCE COUNCIL (TW) 2002-11-12 US disclosed