SCHEMBL7669359

SCHEMBL7669359

CC(C=CC(F)=C(C)c1ccc2c(c1)c(C)c(C)n2C(C)C)=CC(=O)O

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPARG P37231 10/20 0.39
RXRA P19793 6/20 0.39
RXRB P28702 6/20 0.39
RXRG P48443 5/20 0.39
RARA P10276 4/20 0.39
RARB P10826 4/20 0.39
KDM4E B2RXH2 2/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 3/20 0.33
TP53 P04637 2/20 0.33
ATM Q13315 1/20 0.32
ALDH1A1 P00352 1/20 0.31
PKM P14618 1/20 0.31
HTT P42858 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7669355 1.00 PPARG (0.39) PPARGRXRARXRBRXRGRARA
SCHEMBL7675175 0.82 GAA (0.36) PPARGKDM4EGAAMAPTTP53
SCHEMBL7675170 0.82 GAA (0.36) PPARGKDM4EGAAMAPTTP53
SCHEMBL7667150 0.82 RXRA (0.37) PPARGRXRARXRBRXRGRARA
SCHEMBL7667153 0.82 RXRA (0.37) PPARGRXRARXRBRXRGRARA
SCHEMBL7668653 0.79 GAA (0.41) PPARGKDM4EGAAMAPTTP53
SCHEMBL7668646 0.79 GAA (0.41) PPARGKDM4EGAAMAPTTP53
SCHEMBL7667024 0.76 PPARG (0.38) PPARGRXRARXRBRXRGRARA
SCHEMBL7667016 0.76 PPARG (0.38) PPARGRXRARXRBRXRGRARA
SCHEMBL7665546 0.75 ALDH1A1 (0.46) PPARGKDM4EGAAMAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420363-B1 Mono- or polyenic carboxylic acid derivatives EISAI CO., LTD. (JP) 2002-07-16 US disclosed
US-6291508-B1 POTENT ABILITY TO BIND TO RETINOIC ACID RECEPTORS THUS USEFUL IN TREATING PSORIASIS AND RHEUMATOID ARTHRITIS. EISAI CO., LTD. (JP) 2001-09-18 US disclosed
US-6133283-A Mono- or polyenic carboxylic acid derivatives EISAI CO., LTD. (JP) 2000-10-17 US disclosed
US-6030964-A BINDS TO RETINOIC ACID RECEPTORS AND USEFUL FOR TREATING PSORIASIS, AUTOIMMUNE DISEASES, TUMORS, RHEUMATOID ARTHRITIS AND FOR INDUCING IMMUNOSUPPRESSION IN ORGAN TRANSPLANTATION EISAI CO., LTD. (JP) 2000-02-29 US disclosed
US-5977125-A Mono-or polyenic carboxylic acid derivatives EISAI CO., LTD. (JP) 1999-11-02 US disclosed
EP-0790228-A1 MONO- OR POLYENIC CARBOXYLIC ACID DERIVATIVE Eisai Co., Ltd. (JP) 1997-08-20 EP disclosed