SCHEMBL7670604

SCHEMBL7670604

Nc1cccc(C(=O)Nc2ccc(S(=O)(=O)NCC(=O)O)cc2)c1

nearest known ligand 0.74

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.56
MMP2 P08253 1/20 0.54
MMP14 P50281 1/20 0.54
PTGS1 P23219 1/20 0.53
PRMT1 Q99873 1/20 0.52
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
MMP1 P03956 1/20 0.50
GAA P10253 1/20 0.50
MMP12 P39900 1/20 0.50
ALDH1A1 P00352 1/20 0.50
GPR17 Q13304 1/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7673888 0.86 LMNA (0.57) LMNAMMP2MMP14HDAC8HDAC6
SCHEMBL4834530 0.86 LMNA (0.74) LMNAPRMT1MMP1GAAMMP12
SCHEMBL7670709 0.85 GPR17 (0.66) LMNAALDH1A1GPR17MEN1KMT2A
SCHEMBL7670533 0.85 MAPT (0.66) LMNAPRMT1GAAGPR17MEN1
SCHEMBL7665938 0.85 MEN1 (0.66) LMNAMMP2MMP14GAAMEN1
SCHEMBL7670605 0.85 CA1 (0.63) LMNAMMP2MMP14PRMT1ALDH1A1
SCHEMBL25926127 0.82 KMT2A (0.68) PRMT1HDAC8HDAC6ALDH1A1MEN1
SCHEMBL4825269 0.82 MEN1 (0.68) LMNAGAAALDH1A1GPR17MEN1
SCHEMBL7668838 0.82 LMNA (0.68) LMNAMMP2GAAALDH1A1MEN1
SCHEMBL14534186 0.82 MMP1 (0.71) LMNAMMP2MMP14PRMT1MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403644-B1 FOR PREVENTION AND/OR TREATMENT OF DISEASES INDUCED BY OVEREXPRESSION AND EXCESS ACTIVITY OF MATRIX METALLOPROTEINASE; FOR EXAMPLE, RHEUMATOID, ARTHROSTEITIS, UNUSUAL BONE RESORPTION, OSTEOPOROSIS, PERIODONTITIS ONO PHARMACEUTICAL CO., LTD. (JP) 2002-06-11 US claimed
EP-0757037-A2 Sulfonylamino acid derivatives as metalloproteinase inhibitors ONO PHARMACEUTICAL CO., LTD. (JP) 1997-02-05 EP claimed
US-6403644-B1 FOR PREVENTION AND/OR TREATMENT OF DISEASES INDUCED BY OVEREXPRESSION AND EXCESS ACTIVITY OF MATRIX METALLOPROTEINASE; FOR EXAMPLE, RHEUMATOID, ARTHROSTEITIS, UNUSUAL BONE RESORPTION, OSTEOPOROSIS, PERIODONTITIS ONO PHARMACEUTICAL CO., LTD. (JP) 2002-06-11 US disclosed
US-6177466-B1 Sulfonylamino acid derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 2001-01-23 US disclosed
EP-0757037-A2 Sulfonylamino acid derivatives as metalloproteinase inhibitors ONO PHARMACEUTICAL CO., LTD. (JP) 1997-02-05 EP disclosed