SCHEMBL7675309

SCHEMBL7675309

CCOC(Cc1ccccc1)=C(CBr)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
KMT2A Q03164 2/20 0.40
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
AKR1B1 P15121 1/20 0.40
PAM P19021 1/20 0.40
MEN1 O00255 1/20 0.40
TSHR P16473 2/20 0.40
MAPK8 P45983 1/20 0.39
MAPK9 P45984 1/20 0.39
MAPK10 P53779 1/20 0.39
PPID Q08752 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MMP8 P22894 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28728818 0.79 L3MBTL1 (0.42) ALDH1A1L3MBTL1MAPK1SMN1; SMN2KMT2A
SCHEMBL11830681 0.79 ALDH1A1 (0.46) ALDH1A1L3MBTL1MAPK1SMN1; SMN2KMT2A
SCHEMBL4825672 0.79 ALDH1A1 (0.46) ALDH1A1L3MBTL1MAPK1SMN1; SMN2KMT2A
SCHEMBL7672215 0.78 PPID (0.42) ALDH1A1L3MBTL1MAPK1SMN1; SMN2KMT2A
SCHEMBL28757779 0.76 MEN1 (0.49) ALDH1A1L3MBTL1MAPK1SMN1; SMN2KMT2A
SCHEMBL15170431 0.76 MEN1 (0.49) ALDH1A1L3MBTL1MAPK1SMN1; SMN2KMT2A
SCHEMBL112999 0.72 ALDH1A1 (0.68) ALDH1A1L3MBTL1MAPK1SMN1; SMN2KMT2A
SCHEMBL1873977 0.72 ALDH1A1 (0.68) ALDH1A1L3MBTL1MAPK1SMN1; SMN2KMT2A
Benzene SCHEMBL28160801 0.72 ALDH1A1 (0.68) ALDH1A1L3MBTL1MAPK1SMN1; SMN2KMT2A
SCHEMBL1332625 0.72 ALDH1A1 (0.68) ALDH1A1L3MBTL1MAPK1SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0745621-B1 Polymerisable composition based on thio(meth)acrylate monomer, transparent polymer compositions and their optical use ESSILOR INT (FR) 1998-04-15 EP claimed
EP-0745621-A1 Polymerisable composition based on thio(meth)acrylate monomer, transparent polymer compositions and their optional use ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 1996-12-04 EP claimed
US-11752713-B2 Polymer composition and methods using said polymer composition to manufacture ophthalmic lens ESSILOR INTERNATIONAL (FR) 2023-09-12 US disclosed
EP-4235273-A2 ADDITIVE MANUFACTURING PROCESSES FOR TRANSPARENT OPHTHALMIC LENS Essilor International (FR) 2023-08-30 EP disclosed
EP-3027396-B1 ADDITIVE MANUFACTURING PROCESSES FOR TRANSPARENT OPHTHALMIC LENS ESSILOR INT (FR) 2023-06-14 EP disclosed
EP-3027397-B1 ADDITIVE MANUFACTURING FOR TRANSPARENT OPHTHALMIC LENS ESSILOR INT (FR) 2021-07-14 EP disclosed
US-20210072425-A1 Polymer Composition and Methods Using Said Polymer Composition to Manufacture Ophthalmic Lens ESSILOR INTERNATIONAL (FR) 2021-03-11 US disclosed
US-9969135-B2 Additive manufacturing for transparent ophthalmic lens ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2018-05-15 US disclosed
EP-3084484-B1 POLYMER COMPOSITION AND METHODS USING SAID POLYMER COMPOSITION TO MANUFACTURE OPHTHALMIC LENS ESSILOR INT (FR) 2018-03-21 EP disclosed
US-20170031059-A1 Polymer Composition and Methods Using Said Polymer Composition to Manufacture Ophthalmic Lens ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2017-02-02 US disclosed
EP-3084484-A1 POLYMER COMPOSITION AND METHODS USING SAID POLYMER COMPOSITION TO MANUFACTURE OPHTHALMIC LENS Essilor International (Compagnie Générale D'Optique) (FR) 2016-10-26 EP disclosed
US-20160167299-A1 ADDITIVE MANUFACTURING FOR TRANSPARENT OPHTHALMIC LENS ESSILOR INTERNATIONAL (FR) 2016-06-16 US disclosed
EP-3027397-A1 ADDITIVE MANUFACTURING FOR TRANSPARENT OPHTHALMIC LENS Essilor International (Compagnie Générale D'Optique) (FR) 2016-06-08 EP disclosed
EP-3027396-A1 ADDITIVE MANUFACTURING PROCESSES FOR TRANSPARENT OPHTHALMIC LENS Essilor International (Compagnie Générale D'Optique) (FR) 2016-06-08 EP disclosed
US-6472488-B2 MONOMERS CONTAIN THIO-CONTAINING HETEROCYCLES; USE IN MANUFACTURE OF WAVEGUIDES, OPTICAL FIBERS AND SPECTACLE LENSES ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 2002-10-29 US disclosed
US-6307062-B1 E.G., METHACRYLIC ESTER OF 1,4-DITHIACYCLOHEPTANE ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 2001-10-23 US disclosed
EP-0901486-B1 NOVEL (THIO)(METH)ACRYLATE MONOMERS, INTERMEDIATE COMPOUNDS FOR THE SYNTHESIS OF THESE MONOMERS, POLYMERISABLE COMPOSITIONS AND RESULTING POLYMERS AND OPTICAL AND OPHTHALMOLOGIC APPLICATIONS THEREOF ESSILOR INT (FR) 2001-09-26 EP disclosed
EP-0901486-A1 NOVEL (THIO)(METH)ACRYLATE MONOMERS, INTERMEDIATE COMPOUNDS FOR THE SYNTHESIS OF THESE MONOMERS, POLYMERISABLE COMPOSITIONS AND RESULTING POLYMERS AND OPTICAL AND OPHTHALMOLOGIC APPLICATIONS THEREOF ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 1999-03-17 EP disclosed
WO-1998035955-A1 NOVEL (THIO)(METH)ACRYLATE MONOMERS, INTERMEDIATE COMPOUNDS FOR THE SYNTHESIS OF THESE MONOMERS, POLYMERISABLE COMPOSITIONS AND RESULTING POLYMERS AND OPTICAL AND OPHTHALMOLOGIC APPLICATIONS THEREOF ESSILOR INTERNATIONAL - COMPAGNIE GENERALE D'OPTIQUE (FR) 1998-08-20 WO disclosed
EP-0745621-A1 Polymerisable composition based on thio(meth)acrylate monomer, transparent polymer compositions and their optional use ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 1996-12-04 EP disclosed