SCHEMBL7675310

SCHEMBL7675310

CC(=COC(CBr)Cc1ccccc1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPI P09923 1/20 0.41
PKM P14618 1/20 0.41
PTGS1 P23219 1/20 0.41
XIAP P98170 1/20 0.41
SLC7A5 Q01650 1/20 0.41
CYP2C9 P11712 1/20 0.41
CTSK P43235 3/20 0.40
CYP1A2 P05177 1/20 0.40
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
CPA1 P15085 1/20 0.39
AKR1C3 P42330 1/20 0.39
SRR Q9GZT4 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
CTRB1 P17538 3/20 0.38
HPGD P15428 1/20 0.38
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8921434 0.78 ALDH1A1 (0.46) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL106764 0.74 EPHX1 (0.44) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL7672216 0.73 AKR1C3 (0.42) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL29038863 0.72 CYP2C9 (0.38) CYP2C9NPC1RAB9AHPGDALDH1A1
SCHEMBL29038865 0.72 CYP2C9 (0.38) CYP2C9NPC1RAB9AHPGDALDH1A1
SCHEMBL28431910 0.71 SRR (0.46) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL981849 0.70 ALDH1A1 (0.53) CYP2C9AKR1C3NPC1RAB9AHPGD
SCHEMBL2808822 0.70 ALDH1A1 (0.53) CYP2C9AKR1C3NPC1RAB9AHPGD
SCHEMBL9338801 0.70 AKR1C3 (0.46) CYP2C9AKR1C3HPGDALDH1A1
SCHEMBL28474427 0.69 NPC1 (0.47) ALPIPKMPTGS1XIAPSLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0745621-B1 Polymerisable composition based on thio(meth)acrylate monomer, transparent polymer compositions and their optical use ESSILOR INT (FR) 1998-04-15 EP claimed
EP-0745621-A1 Polymerisable composition based on thio(meth)acrylate monomer, transparent polymer compositions and their optional use ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 1996-12-04 EP claimed
US-11752713-B2 Polymer composition and methods using said polymer composition to manufacture ophthalmic lens ESSILOR INTERNATIONAL (FR) 2023-09-12 US disclosed
EP-4235273-A2 ADDITIVE MANUFACTURING PROCESSES FOR TRANSPARENT OPHTHALMIC LENS Essilor International (FR) 2023-08-30 EP disclosed
EP-3027396-B1 ADDITIVE MANUFACTURING PROCESSES FOR TRANSPARENT OPHTHALMIC LENS ESSILOR INT (FR) 2023-06-14 EP disclosed
EP-3027397-B1 ADDITIVE MANUFACTURING FOR TRANSPARENT OPHTHALMIC LENS ESSILOR INT (FR) 2021-07-14 EP disclosed
US-20210072425-A1 Polymer Composition and Methods Using Said Polymer Composition to Manufacture Ophthalmic Lens ESSILOR INTERNATIONAL (FR) 2021-03-11 US disclosed
US-9969135-B2 Additive manufacturing for transparent ophthalmic lens ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2018-05-15 US disclosed
EP-3084484-B1 POLYMER COMPOSITION AND METHODS USING SAID POLYMER COMPOSITION TO MANUFACTURE OPHTHALMIC LENS ESSILOR INT (FR) 2018-03-21 EP disclosed
US-20170031059-A1 Polymer Composition and Methods Using Said Polymer Composition to Manufacture Ophthalmic Lens ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2017-02-02 US disclosed
EP-3084484-A1 POLYMER COMPOSITION AND METHODS USING SAID POLYMER COMPOSITION TO MANUFACTURE OPHTHALMIC LENS Essilor International (Compagnie Générale D'Optique) (FR) 2016-10-26 EP disclosed
US-20160167299-A1 ADDITIVE MANUFACTURING FOR TRANSPARENT OPHTHALMIC LENS ESSILOR INTERNATIONAL (FR) 2016-06-16 US disclosed
EP-3027397-A1 ADDITIVE MANUFACTURING FOR TRANSPARENT OPHTHALMIC LENS Essilor International (Compagnie Générale D'Optique) (FR) 2016-06-08 EP disclosed
EP-3027396-A1 ADDITIVE MANUFACTURING PROCESSES FOR TRANSPARENT OPHTHALMIC LENS Essilor International (Compagnie Générale D'Optique) (FR) 2016-06-08 EP disclosed
US-6472488-B2 MONOMERS CONTAIN THIO-CONTAINING HETEROCYCLES; USE IN MANUFACTURE OF WAVEGUIDES, OPTICAL FIBERS AND SPECTACLE LENSES ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 2002-10-29 US disclosed
US-6307062-B1 E.G., METHACRYLIC ESTER OF 1,4-DITHIACYCLOHEPTANE ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 2001-10-23 US disclosed
EP-0901486-B1 NOVEL (THIO)(METH)ACRYLATE MONOMERS, INTERMEDIATE COMPOUNDS FOR THE SYNTHESIS OF THESE MONOMERS, POLYMERISABLE COMPOSITIONS AND RESULTING POLYMERS AND OPTICAL AND OPHTHALMOLOGIC APPLICATIONS THEREOF ESSILOR INT (FR) 2001-09-26 EP disclosed
EP-0901486-A1 NOVEL (THIO)(METH)ACRYLATE MONOMERS, INTERMEDIATE COMPOUNDS FOR THE SYNTHESIS OF THESE MONOMERS, POLYMERISABLE COMPOSITIONS AND RESULTING POLYMERS AND OPTICAL AND OPHTHALMOLOGIC APPLICATIONS THEREOF ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 1999-03-17 EP disclosed
WO-1998035955-A1 NOVEL (THIO)(METH)ACRYLATE MONOMERS, INTERMEDIATE COMPOUNDS FOR THE SYNTHESIS OF THESE MONOMERS, POLYMERISABLE COMPOSITIONS AND RESULTING POLYMERS AND OPTICAL AND OPHTHALMOLOGIC APPLICATIONS THEREOF ESSILOR INTERNATIONAL - COMPAGNIE GENERALE D'OPTIQUE (FR) 1998-08-20 WO disclosed
EP-0745621-A1 Polymerisable composition based on thio(meth)acrylate monomer, transparent polymer compositions and their optional use ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 1996-12-04 EP disclosed