SCHEMBL7676958

SCHEMBL7676958

O=C(O)C1(C2NCCc3c2[nH]c2ccccc32)CCC1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 2/20 0.60
HTR7 P34969 4/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C19 P33261 1/20 0.53
GRIN2B Q13224 1/20 0.49
PRMT5 O14744 3/20 0.48
EGFR P00533 3/20 0.48
DRD2 P14416 1/20 0.46
SIRT1 Q96EB6 2/20 0.46
SIRT2 Q8IXJ6 1/20 0.46
BRD3 Q15059 1/20 0.45
ABCB1 P08183 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7854266 0.87 CDC42 (0.47) MAPKAPK2SIRT1
SCHEMBL7851653 0.85 MAPKAPK2 (0.62) MAPKAPK2SIRT1
SCHEMBL7676904 0.84 SIRT1 (0.43) MAPKAPK2SIRT1SIRT2
SCHEMBL7680354 0.84 HTR2A (0.47) MAPKAPK2CYP2D6SIRT1
SCHEMBL7680308 0.84 MAPKAPK2 (0.63) MAPKAPK2SIRT1SIRT2
SCHEMBL7843811 0.84 MAPKAPK2 (0.63) MAPKAPK2BRD3
SCHEMBL7680950 0.84 SIRT1 (0.54) MAPKAPK2SIRT1SIRT2
Hydrochloric Acid SCHEMBL7673540 0.83 HTR2A (0.49) MAPKAPK2CYP2D6SIRT1
Hydrochloric Acid SCHEMBL7673537 0.83 HTR2A (0.49) MAPKAPK2CYP2D6SIRT1
Hydrochloric Acid SCHEMBL7678941 0.82 MAPKAPK2 (0.48) MAPKAPK2HTR7CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350757-B1 Beta-carboline compounds LES LABORATOIRES SERVIER (FR) 2002-02-26 US disclosed
EP-1070716-A1 Beta-carboline derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 2001-01-24 EP disclosed